Human GPCR Panel Assay

We provide reliable and comprehensive human GPCR panel assay services on our proprietary functional assay platform (international patent application filed). Our panel services include
  • FlexPanel48, two types of focused panels with 48 GPCRs and
  • large-scale comprehensive panels covering as many as 297 GPCRs.
Listed at the bottom are the 202 non-orphan GPCRs and the 95 orphan GPCRs eligible for panel assays and the 48 GPCRs in each of FlexPanel48 Therapeutic Area Panels. Contact us for details and quotations. flowchart

FlexPanel48
, focused GPCR panels

FlexPanel48 is reasonable small-scale panels with 48 receptors and consists of custom panels and therapeutic area panels.

FlexPanel48 Custom Panels

  • One can choose 48 receptors from the 202 non-orphan GPCRs and the 95 orphan GPCRs on our list.
  • Two assay modes, the agonist and antagonist modes, are available.
    Orphan GPCRs are assayed in the agonist mode only.
  • The two assay modes may coexist in a single panel.

FlexPanel48 Therapeutic Area Panels

Thirteen Therapeutic Areas

  • Immunology/Infection
  • Oncology
  • Hematology
  • Endocrinology/Metabolism
  • Psychiatry
  • Neurology
  • Ophthalmology
  • Cardiology
  • Respiratory
  • Gastrointestinal
  • Dermatology
  • Musculoskeletal
  • Urology/Reproduction
  • Assorted are the 48 GPCRs with high disease-gene association scores according to the DisGeNET database.
  • The receptors in each panel are listed below.
  • Two assay modes, the agonist and antagonist modes, are available.
  • The two assay modes may coexist in a single panel.
  • One can customize a Therapeutic Area Panel by replacing receptors on the list with those of his/her choice.

Panel Assay Examples

FlexPanel48 Endocrinology/Metabolism Panel

TAK875 vs FlexPanel48 Metabol/Endocrinol
Figure 1. TAK-875 screened in the endocrinology/metabolism panel
TAK875 Concentration-response curve
Figure 2. Concentration-response curve for TAK-875
TAK-875, a Phase 3 antidiabetic, was screened in the agonist mode in the FlexPanel48 Endocrinology/Metabolism Panel (Figure 1). TAK-875 selectively activated free fatty acid receptor 1 (FFAR1). Next, TAK-875 was shown to activate FFAR1 in a concentration-dependent manner (Figure 2).
Endocrinology/Metabolism Panel Receptors
1HTR2A11CALCR21FFAR131KISS1R41PTH1R
2HTR2C12CASR22GHSR32S1PR242PROKR2
3CHRM213CNR123GHRHR33MC1R43PTGER4
4CHRM314CCR524GIPR34MC2R44SSTR1
5ADRA1A15CXCR425GLP1R35MC4R45SSTR2
6ADRB116CCKAR26GCGR36MTNR1B46TACR3
7ADRB217CCKBR27FSHR37NPY1R47TRHR
8ADRB318DRD228LHCGR38NPY2R48AVPR2
9AGTR119EDNRA29TSHR39NPY5R
10BRS320EDNRB30GNRHR40OPRM1

FlexPanel48 Psychiatry Panel

Figure 3. Naloxone screened in the psychiatry panel
Figure 4. Concentration-response curves for naloxone
Naloxone, the opioid reversal drug, was screened in the antagonist mode in the FlexPanel48 Psychiatry Panel (Figure 3). Naloxone selectively antagonized opiate receptors OPRD1, OPRK1, and OPRM1. Next, naloxone was shown to antagonize the three opiate receptors in a concentration-dependent manner (Figure 4).
Psychiatry Panel Receptors
1HTR1A11CHRM421CCKBR31HRH141OPRK1
2HTR1B12CHRM522CRHR132HRH242OPRM1
3HTR2A13ADORA2A23CRHR233HRH343OPRL1
4HTR2C14ADRA2A24DRD134GRM244HCRTR1
5HTR5A15ADRA2B25DRD235GRM845TACR1
6HTR616ADRB126DRD336NPSR146AVPR1A
7HTR717ADRB227DRD437NPY1R47OXTR
8CHRM118GRPR28DRD538NPY2R48ADCYAP1R1
9CHRM219CNR129EDNRA39NTSR1
10CHRM320CCKAR30GABBR1/240OPRD1

Large-Scale Comprehensive Panels

Our large-scale panel assays allow comprehensive screening for up to 202 non-orphan GPCRs and 95 orphan GPCRs. The total of 297 GPCRs amenable to panel assays are listed below.

Panel Assay Example

Figure 5. Carvedilol screened for 200 non-orphan GPCRs.
CarvedilolDR_sizeadjusted
Figure 6. Concentration-response curves for carvedilol

Carvedilol, an anti-hypertensive agent, was screened in the antagonist mode for 200 non-orphan GPCRs (Figure 5). Carvedilol selectively antagonized α1A, α1B, α1D, β1, and β2 adrenoceptors. Next, carvedilol was shown to antagonize the above receptors in a concentration-dependent manner (Figure 6).

Panel Receptors

  • Listed are the total of 297 GPCRs amenable to panel assays and the GPCRs in the therapeutic area panels
  • One can customize therapeutic area panels.
All GPCRsImmunology/InfectionOncologyHematologyEndocrinology/MetabolismPsychiatryNeurologyOphthalmologyCardiologyRespiratoryGastrointestinalDermatologyMusculoskeletalUrology/Reproduction
SymbolHGNC nameFamily
HTR1A5-hydroxytryptamine receptor 1A5-Hydroxytryptamine receptors
HTR1B5-hydroxytryptamine receptor 1B5-Hydroxytryptamine receptors
HTR1D5-hydroxytryptamine receptor 1D5-Hydroxytryptamine receptors
HTR1E5-hydroxytryptamine receptor 1E5-Hydroxytryptamine receptors
HTR1F5-hydroxytryptamine receptor 1F5-Hydroxytryptamine receptors
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptors
HTR2B5-hydroxytryptamine receptor 2B5-Hydroxytryptamine receptors
HTR2C5-hydroxytryptamine receptor 2C5-Hydroxytryptamine receptors
HTR45-hydroxytryptamine receptor 45-Hydroxytryptamine receptors
HTR5A5-hydroxytryptamine receptor 5A5-Hydroxytryptamine receptors
HTR65-hydroxytryptamine receptor 65-Hydroxytryptamine receptors
HTR75-hydroxytryptamine receptor 75-Hydroxytryptamine receptors
CHRM1cholinergic receptor muscarinic 1Acetylcholine receptors (muscarinic)
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
CHRM4cholinergic receptor muscarinic 4Acetylcholine receptors (muscarinic)
CHRM5cholinergic receptor muscarinic 5Acetylcholine receptors (muscarinic)
ADORA1adenosine A1 receptorAdenosine receptors
ADORA2Aadenosine A2a receptorAdenosine receptors
ADORA2Badenosine A2b receptorAdenosine receptors
ADORA3adenosine A3 receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA1Badrenoceptor alpha 1BAdrenoceptors
ADRA1Dadrenoceptor alpha 1DAdrenoceptors
ADRA2Aadrenoceptor alpha 2AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRA2Cadrenoceptor alpha 2CAdrenoceptors
ADRB1adrenoceptor beta 1Adrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
ADRB3adrenoceptor beta 3Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
APLNRapelin receptorApelin receptor
GPBAR1G protein-coupled bile acid receptor 1Bile acid receptor
BRS3bombesin receptor subtype 3Bombesin receptors
GRPRgastrin releasing peptide receptorBombesin receptors
NMBRneuromedin B receptorBombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CALCRLcalcitonin receptor like receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
GPR55G protein-coupled receptor 55Cannabinoid receptors
GPR119G protein-coupled receptor 119Cannabinoid receptors
CMKLR1chemerin chemokine-like receptor 1Chemerin receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CCR8C-C motif chemokine receptor 8Chemokine receptors
CCR9C-C motif chemokine receptor 9Chemokine receptors
CCR10C-C motif chemokine receptor 10Chemokine receptors
CXCR1C-X-C motif chemokine receptor 1Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
XCR1X-C motif chemokine receptor 1Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
CCKARcholecystokinin A receptorCholecystokinin receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
C3AR1complement C3a receptor 1Complement peptide receptors
C5AR1complement C5a receptor 1Complement peptide receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
CRHR2corticotropin releasing hormone receptor 2Corticotropin-releasing factor receptors
DRD1dopamine receptor D1Dopamine receptors
DRD2dopamine receptor D2Dopamine receptors
DRD3dopamine receptor D3Dopamine receptors
DRD4dopamine receptor D4Dopamine receptors
DRD5dopamine receptor D5Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GPR183G protein-coupled receptor 183Steroid receptors
FPR1formyl peptide receptor 1Formylpeptide receptors
FPR2formyl peptide receptor 2Formylpeptide receptors
FPR3formyl peptide receptor 3Formylpeptide receptors
FFAR1free fatty acid receptor 1Free fatty acid receptors
FFAR3free fatty acid receptor 3Free fatty acid receptors
GPR84G protein-coupled receptor 84Free fatty acid receptors
FFAR4free fatty acid receptor 4Free fatty acid receptors
GABBR1gamma-aminobutyric acid type B receptor subunit 1GABAB receptors
GABBR2gamma-aminobutyric acid type B receptor subunit 2GABAB receptors
GALR1galanin receptor 1Galanin receptors
GALR2galanin receptor 2Galanin receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GHRHRgrowth hormone releasing hormone receptorGlucagon receptor family
GIPRgastric inhibitory polypeptide receptorGlucagon receptor family
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
GLP2Rglucagon like peptide 2 receptorGlucagon receptor family
GCGRglucagon receptorGlucagon receptor family
SCTRsecretin receptorGlucagon receptor family
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptors
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptors
HRH1histamine receptor H1Histamine receptors
HRH2histamine receptor H2Histamine receptors
HRH3histamine receptor H3Histamine receptors
HRH4histamine receptor H4Histamine receptors
HCAR2hydroxycarboxylic acid receptor 2Hydroxycarboxylic acid receptors
HCAR3hydroxycarboxylic acid receptor 3Hydroxycarboxylic acid receptors
KISS1RKISS1 receptorKisspeptin receptor
LTB4Rleukotriene B4 receptorLeukotriene receptors
LTB4R2leukotriene B4 receptor 2Leukotriene receptors
CYSLTR1cysteinyl leukotriene receptor 1Leukotriene receptors
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptors
OXER1oxoeicosanoid receptor 1Leukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
LPAR3lysophosphatidic acid receptor 3Lysophospholipid (LPA) receptors
LPAR4lysophosphatidic acid receptor 4Lysophospholipid (LPA) receptors
LPAR5lysophosphatidic acid receptor 5Lysophospholipid (LPA) receptors
LPAR6lysophosphatidic acid receptor 6Lysophospholipid (LPA) receptors
S1PR1sphingosine-1-phosphate receptor 1Lysophospholipid (S1P) receptors
S1PR2sphingosine-1-phosphate receptor 2Lysophospholipid (S1P) receptors
S1PR3sphingosine-1-phosphate receptor 3Lysophospholipid (S1P) receptors
S1PR5sphingosine-1-phosphate receptor 5Lysophospholipid (S1P) receptors
MCHR1melanin concentrating hormone receptor 1Melanin-concentrating hormone receptors
MCHR2melanin concentrating hormone receptor 2Melanin-concentrating hormone receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
MC2Rmelanocortin 2 receptorMelanocortin receptors
MC3Rmelanocortin 3 receptorMelanocortin receptors
MC4Rmelanocortin 4 receptorMelanocortin receptors
MC5Rmelanocortin 5 receptorMelanocortin receptors
MTNR1Amelatonin receptor 1AMelatonin receptors
MTNR1Bmelatonin receptor 1BMelatonin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
GRM2glutamate metabotropic receptor 2Metabotropic glutamate receptors
GRM4glutamate metabotropic receptor 4Metabotropic glutamate receptors
GRM6glutamate metabotropic receptor 6Metabotropic glutamate receptors
GRM8glutamate metabotropic receptor 8Metabotropic glutamate receptors
MLNRmotilin receptorMotilin receptor
NMUR1neuromedin U receptor 1Neuromedin U receptors
NMUR2neuromedin U receptor 2Neuromedin U receptors
NPFFR1neuropeptide FF receptor 1Neuropeptide FF/neuropeptide AF receptors
NPFFR2neuropeptide FF receptor 2Neuropeptide FF/neuropeptide AF receptors
NPSR1neuropeptide S receptor 1Neuropeptide S receptor
NPBWR1neuropeptides B and W receptor 1Neuropeptide W/neuropeptide B receptors
NPBWR2neuropeptides B and W receptor 2Neuropeptide W/neuropeptide B receptors
NPY1Rneuropeptide Y receptor Y1Neuropeptide Y receptors
NPY2Rneuropeptide Y receptor Y2Neuropeptide Y receptors
NPY4Rneuropeptide Y receptor Y4Neuropeptide Y receptors
NPY5Rneuropeptide Y receptor Y5Neuropeptide Y receptors
NTSR1neurotensin receptor 1Neurotensin receptors
NTSR2neurotensin receptor 2Neurotensin receptors
OPRD1opioid receptor delta 1Opioid receptors
OPRK1opioid receptor kappa 1Opioid receptors
OPRM1opioid receptor mu 1Opioid receptors
OPRL1opioid related nociceptin receptor 1Opioid receptors
HCRTR1hypocretin receptor 1Orexin receptors
HCRTR2hypocretin receptor 2Orexin receptors
OXGR1oxoglutarate receptor 1Oxoglutarate receptors
P2RY1purinergic receptor P2Y1P2Y receptors
P2RY2purinergic receptor P2Y2P2Y receptors
P2RY4pyrimidinergic receptor P2Y4P2Y receptors
P2RY6pyrimidinergic receptor P2Y6P2Y receptors
P2RY11purinergic receptor P2Y11P2Y receptors
P2RY12purinergic receptor P2Y12P2Y receptors
P2RY13purinergic receptor P2Y13P2Y receptors
P2RY14purinergic receptor P2Y14P2Y receptors
P2RY10P2Y receptor family member 10P2Y receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PTH2Rparathyroid hormone 2 receptorParathyroid hormone receptors
PROKR1prokineticin receptor 1Prokineticin receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PRLHRprolactin releasing hormone receptorProlactin-releasing peptide receptor
PTGDRprostaglandin D2 receptorProstanoid receptors
PTGDR2prostaglandin D2 receptor 2Prostanoid receptors
PTGER1prostaglandin E receptor 1Prostanoid receptors
PTGER2prostaglandin E receptor 2Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
PTGFRprostaglandin F receptorProstanoid receptors
PTGIRprostaglandin I2 receptorProstanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
F2RL2coagulation factor II thrombin receptor like 2Proteinase-activated receptors
F2RL3F2R like thrombin or trypsin receptor 3Proteinase-activated receptors
QRFPRpyroglutamylated RFamide peptide receptorQRFP receptor
RXFP1relaxin family peptide receptor 1Relaxin family peptide receptors
RXFP2relaxin family peptide receptor 2Relaxin family peptide receptors
RXFP3relaxin family peptide receptor 3Relaxin family peptide receptors
RXFP4relaxin family peptide/INSL5 receptor 4Relaxin family peptide receptors
SSTR1somatostatin receptor 1Somatostatin receptors
SSTR2somatostatin receptor 2Somatostatin receptors
SSTR3somatostatin receptor 3Somatostatin receptors
SSTR4somatostatin receptor 4Somatostatin receptors
SSTR5somatostatin receptor 5Somatostatin receptors
SUCNR1succinate receptor 1Succinate receptor
TACR1tachykinin receptor 1Tachykinin receptors
TACR2tachykinin receptor 2Tachykinin receptors
TACR3tachykinin receptor 3Tachykinin receptors
TRHRthyrotropin releasing hormone receptorThyrotropin-releasing hormone receptors
TAAR1trace amine associated receptor 1Trace amine receptor
UTS2Rurotensin 2 receptorUrotensin receptor
AVPR1Aarginine vasopressin receptor 1AVasopressin and oxytocin receptors
AVPR1Barginine vasopressin receptor 1BVasopressin and oxytocin receptors
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptors
OXTRoxytocin receptorVasopressin and oxytocin receptors
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptors
VIPR1vasoactive intestinal peptide receptor 1VIP and PACAP receptors
VIPR2vasoactive intestinal peptide receptor 2VIP and PACAP receptors
AGTR2angiotensin II receptor type 2Orphan receptors
GPRC6AG protein-coupled receptor class C group 6 member AOrphan receptors
GPR18G protein-coupled receptor 18Orphan receptors
GPR1G protein-coupled receptor 1Orphan receptors
ACKR4atypical chemokine receptor 4Orphan receptors
CCRL2C-C motif chemokine receptor like 2Orphan receptors
ACKR1atypical chemokine receptor 1 (Duffy blood group)Orphan receptors
ACKR2atypical chemokine receptor 2Orphan receptors
ACKR3atypical chemokine receptor 3Orphan receptors
GPER1G protein-coupled estrogen receptor 1Orphan receptors
GPR151G protein-coupled receptor 151Orphan receptors
TAAR2trace amine associated receptor 2Orphan receptors
TAAR5trace amine associated receptor 5Orphan receptors
TAAR6trace amine associated receptor 6Orphan receptors
TAAR8trace amine associated receptor 8Orphan receptors
TAAR9trace amine associated receptor 9Orphan receptors
GPR4G protein-coupled receptor 4Orphan receptors
GPR65G protein-coupled receptor 65Orphan receptors
GPR68G protein-coupled receptor 68Orphan receptors
GPR132G protein-coupled receptor 132Orphan receptors
GPR3G protein-coupled receptor 3Orphan receptors
GPR6G protein-coupled receptor 6Orphan receptors
GPR12G protein-coupled receptor 12Orphan receptors
GPR15G protein-coupled receptor 15Orphan receptors
GPR17G protein-coupled receptor 17Orphan receptors
GPR19G protein-coupled receptor 19Orphan receptors
GPR20G protein-coupled receptor 20Orphan receptors
GPR21G protein-coupled receptor 21Orphan receptors
GPR22G protein-coupled receptor 22Orphan receptors
GPR25G protein-coupled receptor 25Orphan receptors
GPR26G protein-coupled receptor 26Orphan receptors
GPR27G protein-coupled receptor 27Orphan receptors
GPR31G protein-coupled receptor 31Orphan receptors
GPR32G protein-coupled receptor 32Orphan receptors
GPR34G protein-coupled receptor 34Orphan receptors
GPR35G protein-coupled receptor 35Orphan receptors
GPR37G protein-coupled receptor 37Orphan receptors
GPR37L1G protein-coupled receptor 37 like 1Orphan receptors
GPR39G protein-coupled receptor 39Orphan receptors
GPR45G protein-coupled receptor 45Orphan receptors
GPR50G protein-coupled receptor 50Orphan receptors
GPR52G protein-coupled receptor 52Orphan receptors
GPR61G protein-coupled receptor 61Orphan receptors
GPR62G protein-coupled receptor 62Orphan receptors
GPR63G protein-coupled receptor 63Orphan receptors
GPR75G protein-coupled receptor 75Orphan receptors
GPR78G protein-coupled receptor 78Orphan receptors
GPR82G protein-coupled receptor 82Orphan receptors
GPR83G protein-coupled receptor 83Orphan receptors
GPR85G protein-coupled receptor 85Orphan receptors
GPR87G protein-coupled receptor 87Orphan receptors
GPR88G protein-coupled receptor 88Orphan receptors
GPR101G protein-coupled receptor 101Orphan receptors
GPR135G protein-coupled receptor 135Orphan receptors
GPR139G protein-coupled receptor 139Orphan receptors
GPR141G protein-coupled receptor 141Orphan receptors
GPR142G protein-coupled receptor 142Orphan receptors
GPR146G protein-coupled receptor 146Orphan receptors
GPR148G protein-coupled receptor 148Orphan receptors
GPR149G protein-coupled receptor 149Orphan receptors
GPR150G protein-coupled receptor 150Orphan receptors
GPR152G protein-coupled receptor 152Orphan receptors
GPR153G protein-coupled receptor 153Orphan receptors
GPR160G protein-coupled receptor 160Orphan receptors
GPR161G protein-coupled receptor 161Orphan receptors
GPR162G protein-coupled receptor 162Orphan receptors
GPR171G protein-coupled receptor 171Orphan receptors
GPR173G protein-coupled receptor 173Orphan receptors
GPR174G protein-coupled receptor 174Orphan receptors
GPR176G protein-coupled receptor 176Orphan receptors
GPR182G protein-coupled receptor 182Orphan receptors
LGR4leucine rich repeat containing G protein-coupled receptor 4Orphan receptors
LGR5leucine rich repeat containing G protein-coupled receptor 5Orphan receptors
LGR6leucine rich repeat containing G protein-coupled receptor 6Orphan receptors
MAS1MAS1 proto-oncogene, G protein-coupled receptorOrphan receptors
MAS1LMAS1 proto-oncogene like, G protein-coupled receptorOrphan receptors
MRGPRDMAS related GPR family member DOrphan receptors
MRGPREMAS related GPR family member EOrphan receptors
MRGPRFMAS related GPR family member FOrphan receptors
MRGPRGMAS related GPR family member GOrphan receptors
MRGPRX1MAS related GPR family member X1Orphan receptors
MRGPRX2MAS related GPR family member X2Orphan receptors
MRGPRX3MAS related GPR family member X3Orphan receptors
MRGPRX4MAS related GPR family member X4Orphan receptors
GPR156G protein-coupled receptor 156Orphan receptors
GPR158G protein-coupled receptor 158Orphan receptors
GPRC5AG protein-coupled receptor class C group 5 member AOrphan receptors
GPRC5BG protein-coupled receptor class C group 5 member BOrphan receptors
GPRC5CG protein-coupled receptor class C group 5 member COrphan receptors
GPRC5DG protein-coupled receptor class C group 5 member DOrphan receptors
GPR107G protein-coupled receptor 107Orphan receptors
GPR137G protein-coupled receptor 137Orphan receptors
GPR143G protein-coupled receptor 143Orphan receptors
GPR157G protein-coupled receptor 157Orphan receptors
TPRA1transmembrane protein adipocyte associated 1Orphan receptors
SymbolHGNC nameFamily
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA2Aadenosine A2a receptorAdenosine receptors
ADORA2Badenosine A2b receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CCR8C-C motif chemokine receptor 8Chemokine receptors
CCR9C-C motif chemokine receptor 9Chemokine receptors
CXCR1C-X-C motif chemokine receptor 1Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
C5AR1complement C5a receptor 1Complement peptide receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GPR183G protein-coupled receptor 183Steroid receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
HRH1histamine receptor H1Histamine receptors
LTB4Rleukotriene B4 receptorLeukotriene receptors
CYSLTR1cysteinyl leukotriene receptor 1Leukotriene receptors
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
MC2Rmelanocortin 2 receptorMelanocortin receptors
OPRM1opioid receptor mu 1Opioid receptors
P2RY12purinergic receptor P2Y12P2Y receptors
PTGDR2prostaglandin D2 receptor 2Prostanoid receptors
PTGER2prostaglandin E receptor 2Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptors
SymbolHGNC nameFamily
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
GRPRgastrin releasing peptide receptorBombesin receptors
NMBRneuromedin B receptorBombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CCKARcholecystokinin A receptorCholecystokinin receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptors
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptors
HRH4histamine receptor H4Histamine receptors
KISS1RKISS1 receptorKisspeptin receptor
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptors
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
LPAR3lysophosphatidic acid receptor 3Lysophospholipid (LPA) receptors
S1PR1sphingosine-1-phosphate receptor 1Lysophospholipid (S1P) receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
NTSR1neurotensin receptor 1Neurotensin receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PTGER1prostaglandin E receptor 1Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR1somatostatin receptor 1Somatostatin receptors
SSTR2somatostatin receptor 2Somatostatin receptors
SSTR4somatostatin receptor 4Somatostatin receptors
SymbolHGNC nameFamily
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CCR8C-C motif chemokine receptor 8Chemokine receptors
CCR9C-C motif chemokine receptor 9Chemokine receptors
CCR10C-C motif chemokine receptor 10Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
C5AR1complement C5a receptor 1Complement peptide receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GPR183G protein-coupled receptor 183Steroid receptors
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
CYSLTR1cysteinyl leukotriene receptor 1Leukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
S1PR1sphingosine-1-phosphate receptor 1Lysophospholipid (S1P) receptors
S1PR2sphingosine-1-phosphate receptor 2Lysophospholipid (S1P) receptors
NPY5Rneuropeptide Y receptor Y5Neuropeptide Y receptors
OPRK1opioid receptor kappa 1Opioid receptors
OPRM1opioid receptor mu 1Opioid receptors
P2RY12purinergic receptor P2Y12P2Y receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PTGDRprostaglandin D2 receptorProstanoid receptors
PTGDR2prostaglandin D2 receptor 2Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL3F2R like thrombin or trypsin receptor 3Proteinase-activated receptors
RXFP1relaxin family peptide receptor 1Relaxin family peptide receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptors
VIPR1vasoactive intestinal peptide receptor 1VIP and PACAP receptors
SymbolHGNC nameFamily
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptors
HTR2C5-hydroxytryptamine receptor 2C5-Hydroxytryptamine receptors
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRB1adrenoceptor beta 1Adrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
ADRB3adrenoceptor beta 3Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CCKARcholecystokinin A receptorCholecystokinin receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
FFAR1free fatty acid receptor 1Free fatty acid receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GHRHRgrowth hormone releasing hormone receptorGlucagon receptor family
GIPRgastric inhibitory polypeptide receptorGlucagon receptor family
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
GCGRglucagon receptorGlucagon receptor family
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptors
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptors
KISS1RKISS1 receptorKisspeptin receptor
S1PR2sphingosine-1-phosphate receptor 2Lysophospholipid (S1P) receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
MC2Rmelanocortin 2 receptorMelanocortin receptors
MC4Rmelanocortin 4 receptorMelanocortin receptors
MTNR1Bmelatonin receptor 1BMelatonin receptors
NPY1Rneuropeptide Y receptor Y1Neuropeptide Y receptors
NPY2Rneuropeptide Y receptor Y2Neuropeptide Y receptors
NPY5Rneuropeptide Y receptor Y5Neuropeptide Y receptors
OPRM1opioid receptor mu 1Opioid receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
SSTR1somatostatin receptor 1Somatostatin receptors
SSTR2somatostatin receptor 2Somatostatin receptors
TACR3tachykinin receptor 3Tachykinin receptors
TRHRthyrotropin releasing hormone receptorThyrotropin-releasing hormone receptors
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptors
SymbolHGNC nameFamily
HTR1A5-hydroxytryptamine receptor 1A5-Hydroxytryptamine receptors
HTR1B5-hydroxytryptamine receptor 1B5-Hydroxytryptamine receptors
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptors
HTR2C5-hydroxytryptamine receptor 2C5-Hydroxytryptamine receptors
HTR5A5-hydroxytryptamine receptor 5A5-Hydroxytryptamine receptors
HTR65-hydroxytryptamine receptor 65-Hydroxytryptamine receptors
HTR75-hydroxytryptamine receptor 75-Hydroxytryptamine receptors
CHRM1cholinergic receptor muscarinic 1Acetylcholine receptors (muscarinic)
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
CHRM4cholinergic receptor muscarinic 4Acetylcholine receptors (muscarinic)
CHRM5cholinergic receptor muscarinic 5Acetylcholine receptors (muscarinic)
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA2Aadrenoceptor alpha 2AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB1adrenoceptor beta 1Adrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
GRPRgastrin releasing peptide receptorBombesin receptors
CNR1cannabinoid receptor 1Cannabinoid receptors
CCKARcholecystokinin A receptorCholecystokinin receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
CRHR2corticotropin releasing hormone receptor 2Corticotropin-releasing factor receptors
DRD1dopamine receptor D1Dopamine receptors
DRD2dopamine receptor D2Dopamine receptors
DRD3dopamine receptor D3Dopamine receptors
DRD4dopamine receptor D4Dopamine receptors
DRD5dopamine receptor D5Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
GABBR1/2gamma-aminobutyric acid type B receptor subunits 1/2GABAB receptors
HRH1histamine receptor H1Histamine receptors
HRH2histamine receptor H2Histamine receptors
HRH3histamine receptor H3Histamine receptors
GRM2glutamate metabotropic receptor 2Metabotropic glutamate receptors
GRM8glutamate metabotropic receptor 8Metabotropic glutamate receptors
NPSR1neuropeptide S receptor 1Neuropeptide S receptor
NPY1Rneuropeptide Y receptor Y1Neuropeptide Y receptors
NPY2Rneuropeptide Y receptor Y2Neuropeptide Y receptors
NTSR1neurotensin receptor 1Neurotensin receptors
OPRD1opioid receptor delta 1Opioid receptors
OPRK1opioid receptor kappa 1Opioid receptors
OPRM1opioid receptor mu 1Opioid receptors
OPRL1opioid related nociceptin receptor 1Opioid receptors
HCRTR1hypocretin receptor 1Orexin receptors
TACR1tachykinin receptor 1Tachykinin receptors
AVPR1Aarginine vasopressin receptor 1AVasopressin and oxytocin receptors
OXTRoxytocin receptorVasopressin and oxytocin receptors
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptors
SymbolHGNC nameFamily
HTR1A5-hydroxytryptamine receptor 1A5-Hydroxytryptamine receptors
HTR1B5-hydroxytryptamine receptor 1B5-Hydroxytryptamine receptors
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptors
HTR2C5-hydroxytryptamine receptor 2C5-Hydroxytryptamine receptors
HTR75-hydroxytryptamine receptor 75-Hydroxytryptamine receptors
CHRM1cholinergic receptor muscarinic 1Acetylcholine receptors (muscarinic)
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM4cholinergic receptor muscarinic 4Acetylcholine receptors (muscarinic)
ADORA1adenosine A1 receptorAdenosine receptors
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA1Badrenoceptor alpha 1BAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CCR9C-C motif chemokine receptor 9Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
DRD1dopamine receptor D1Dopamine receptors
DRD2dopamine receptor D2Dopamine receptors
DRD3dopamine receptor D3Dopamine receptors
DRD4dopamine receptor D4Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GABBR1/2gamma-aminobutyric acid type B receptor subunits 1/2GABAB receptors
HRH3histamine receptor H3Histamine receptors
KISS1RKISS1 receptorKisspeptin receptor
MC1Rmelanocortin 1 receptorMelanocortin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
NPY1Rneuropeptide Y receptor Y1Neuropeptide Y receptors
NPY2Rneuropeptide Y receptor Y2Neuropeptide Y receptors
OPRK1opioid receptor kappa 1Opioid receptors
OPRM1opioid receptor mu 1Opioid receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER1prostaglandin E receptor 1Prostanoid receptors
SSTR1somatostatin receptor 1Somatostatin receptors
SSTR2somatostatin receptor 2Somatostatin receptors
SSTR3somatostatin receptor 3Somatostatin receptors
SSTR4somatostatin receptor 4Somatostatin receptors
SSTR5somatostatin receptor 5Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
TACR3tachykinin receptor 3Tachykinin receptors
SymbolHGNC nameFamily
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
DRD5dopamine receptor D5Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
FFAR4free fatty acid receptor 4Free fatty acid receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
HCAR2hydroxycarboxylic acid receptor 2Hydroxycarboxylic acid receptors
KISS1RKISS1 receptorKisspeptin receptor
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptors
OXER1oxoeicosanoid receptor 1Leukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
LPAR3lysophosphatidic acid receptor 3Lysophospholipid (LPA) receptors
LPAR6lysophosphatidic acid receptor 6Lysophospholipid (LPA) receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
MTNR1Amelatonin receptor 1AMelatonin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
GRM6glutamate metabotropic receptor 6Metabotropic glutamate receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
PTGFRprostaglandin F receptorProstanoid receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR4somatostatin receptor 4Somatostatin receptors
SUCNR1succinate receptor 1Succinate receptor
TACR3tachykinin receptor 3Tachykinin receptors
VIPR2vasoactive intestinal peptide receptor 2VIP and PACAP receptors
SymbolHGNC nameFamily
HTR1B5-hydroxytryptamine receptor 1B5-Hydroxytryptamine receptors
HTR2B5-hydroxytryptamine receptor 2B5-Hydroxytryptamine receptors
HTR45-hydroxytryptamine receptor 45-Hydroxytryptamine receptors
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA1adenosine A1 receptorAdenosine receptors
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA1Badrenoceptor alpha 1BAdrenoceptors
ADRA2Aadrenoceptor alpha 2AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRA2Cadrenoceptor alpha 2CAdrenoceptors
ADRB1adrenoceptor beta 1Adrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
ADRB3adrenoceptor beta 3Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
APLNRapelin receptorApelin receptor
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
CRHR2corticotropin releasing hormone receptor 2Corticotropin-releasing factor receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
HRH1histamine receptor H1Histamine receptors
HRH3histamine receptor H3Histamine receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
OPRD1opioid receptor delta 1Opioid receptors
OPRK1opioid receptor kappa 1Opioid receptors
OPRM1opioid receptor mu 1Opioid receptors
P2RY1purinergic receptor P2Y1P2Y receptors
P2RY12purinergic receptor P2Y12P2Y receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
TACR1tachykinin receptor 1Tachykinin receptors
UTS2Rurotensin 2 receptorUrotensin receptor
AVPR1Aarginine vasopressin receptor 1AVasopressin and oxytocin receptors
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptors
SymbolHGNC nameFamily
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptors
HTR2B5-hydroxytryptamine receptor 2B5-Hydroxytryptamine receptors
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA1adenosine A1 receptorAdenosine receptors
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR8C-C motif chemokine receptor 8Chemokine receptors
CCR9C-C motif chemokine receptor 9Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
C3AR1complement C3a receptor 1Complement peptide receptors
C5AR1complement C5a receptor 1Complement peptide receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
HRH1histamine receptor H1Histamine receptors
CYSLTR1cysteinyl leukotriene receptor 1Leukotriene receptors
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
NPSR1neuropeptide S receptor 1Neuropeptide S receptor
OPRM1opioid receptor mu 1Opioid receptors
P2RY12purinergic receptor P2Y12P2Y receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PTGDR2prostaglandin D2 receptor 2Prostanoid receptors
PTGER2prostaglandin E receptor 2Prostanoid receptors
PTGFRprostaglandin F receptorProstanoid receptors
PTGIRprostaglandin I2 receptorProstanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
TACR2tachykinin receptor 2Tachykinin receptors
OXTRoxytocin receptorVasopressin and oxytocin receptors
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptors
SymbolHGNC nameFamily
HTR1A5-hydroxytryptamine receptor 1A5-Hydroxytryptamine receptors
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA3adenosine A3 receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB1adrenoceptor beta 1Adrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
GPBAR1G protein-coupled bile acid receptor 1Bile acid receptor
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CXCR1C-X-C motif chemokine receptor 1Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
CCKARcholecystokinin A receptorCholecystokinin receptors
CCKBRcholecystokinin B receptorCholecystokinin receptors
CRHR2corticotropin releasing hormone receptor 2Corticotropin-releasing factor receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
FPR2formyl peptide receptor 2Formylpeptide receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
HRH2histamine receptor H2Histamine receptors
HRH4histamine receptor H4Histamine receptors
KISS1RKISS1 receptorKisspeptin receptor
LTB4Rleukotriene B4 receptorLeukotriene receptors
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
OPRM1opioid receptor mu 1Opioid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
F2RL3F2R like thrombin or trypsin receptor 3Proteinase-activated receptors
SSTR1somatostatin receptor 1Somatostatin receptors
SSTR2somatostatin receptor 2Somatostatin receptors
SSTR3somatostatin receptor 3Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
VIPR1vasoactive intestinal peptide receptor 1VIP and PACAP receptors
SymbolHGNC nameFamily
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Aadrenoceptor alpha 2AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
NMBRneuromedin B receptorBombesin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR4C-C motif chemokine receptor 4Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
HRH1histamine receptor H1Histamine receptors
HRH4histamine receptor H4Histamine receptors
HCAR2hydroxycarboxylic acid receptor 2Hydroxycarboxylic acid receptors
HCAR3hydroxycarboxylic acid receptor 3Hydroxycarboxylic acid receptors
KISS1RKISS1 receptorKisspeptin receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
LPAR6lysophosphatidic acid receptor 6Lysophospholipid (LPA) receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
OPRM1opioid receptor mu 1Opioid receptors
P2RY12purinergic receptor P2Y12P2Y receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER1prostaglandin E receptor 1Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
UTS2Rurotensin 2 receptorUrotensin receptor
SymbolHGNC nameFamily
HTR75-hydroxytryptamine receptor 75-Hydroxytryptamine receptors
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADORA2Aadenosine A2a receptorAdenosine receptors
ADRA2Aadrenoceptor alpha 2AAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CCR1C-C motif chemokine receptor 1Chemokine receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CCR7C-C motif chemokine receptor 7Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR5C-X-C motif chemokine receptor 5Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
C5AR1complement C5a receptor 1Complement peptide receptors
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GABBR1/2gamma-aminobutyric acid type B receptor subunits 1/2GABAB receptors
GHSRgrowth hormone secretagogue receptorGhrelin receptor
GHRHRgrowth hormone releasing hormone receptorGlucagon receptor family
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptors
KISS1RKISS1 receptorKisspeptin receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
MC1Rmelanocortin 1 receptorMelanocortin receptors
MC2Rmelanocortin 2 receptorMelanocortin receptors
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PTH2Rparathyroid hormone 2 receptorParathyroid hormone receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
F2RL1F2R like trypsin receptor 1Proteinase-activated receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR1tachykinin receptor 1Tachykinin receptors
TACR3tachykinin receptor 3Tachykinin receptors
TRHRthyrotropin releasing hormone receptorThyrotropin-releasing hormone receptors
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptors
SymbolHGNC nameFamily
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)
ADRA1Aadrenoceptor alpha 1AAdrenoceptors
ADRA2Badrenoceptor alpha 2BAdrenoceptors
ADRB2adrenoceptor beta 2Adrenoceptors
AGTR1angiotensin II receptor type 1Angiotensin receptors
BRS3bombesin receptor subtype 3Bombesin receptors
GRPRgastrin releasing peptide receptorBombesin receptors
CALCRcalcitonin receptorCalcitonin receptors
CASRcalcium sensing receptorCalcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptors
CMKLR1chemerin chemokine-like receptor 1Chemerin receptors
CCR2C-C motif chemokine receptor 2Chemokine receptors
CCR5C-C motif chemokine receptor 5 (gene/pseudogene)Chemokine receptors
CCR6C-C motif chemokine receptor 6Chemokine receptors
CXCR2C-X-C motif chemokine receptor 2Chemokine receptors
CXCR3C-X-C motif chemokine receptor 3Chemokine receptors
CXCR4C-X-C motif chemokine receptor 4Chemokine receptors
CXCR6C-X-C motif chemokine receptor 6Chemokine receptors
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptors
DRD1dopamine receptor D1Dopamine receptors
DRD2dopamine receptor D2Dopamine receptors
EDNRAendothelin receptor type AEndothelin receptors
EDNRBendothelin receptor type BEndothelin receptors
GLP1Rglucagon like peptide 1 receptorGlucagon receptor family
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptors
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptors
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptors
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptors
KISS1RKISS1 receptorKisspeptin receptor
PTAFRplatelet activating factor receptorPlatelet-activating factor receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptors
MC2Rmelanocortin 2 receptorMelanocortin receptors
MTNR1Bmelatonin receptor 1BMelatonin receptors
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptors
PROKR2prokineticin receptor 2Prokineticin receptors
PTGER1prostaglandin E receptor 1Prostanoid receptors
PTGER2prostaglandin E receptor 2Prostanoid receptors
PTGER4prostaglandin E receptor 4Prostanoid receptors
PTGFRprostaglandin F receptorProstanoid receptors
F2Rcoagulation factor II thrombin receptorProteinase-activated receptors
RXFP1relaxin family peptide receptor 1Relaxin family peptide receptors
RXFP2relaxin family peptide receptor 2Relaxin family peptide receptors
SSTR4somatostatin receptor 4Somatostatin receptors
TACR3tachykinin receptor 3Tachykinin receptors
UTS2Rurotensin 2 receptorUrotensin receptor
AVPR1Aarginine vasopressin receptor 1AVasopressin and oxytocin receptors
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptors

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