ADORA1

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
ADORA1
HGNC name
adenosine A1 receptor
Family
Adenosine receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=18
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Description

Figure. Concentration-dependent activation of ADORA1 by NECA. Reporter cells were transfected with either the expression plasmid for adeno­sine A1 receptor (ADORA1) or the mock plasmid and treated with various concentrations of 5'-N-ethyl­carbox­amido­adeno­sine (NECA). Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 4.8 nM.