GRPR

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
GRPR
HGNC name
gastrin releasing peptide receptor
Family
Bombesin receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=39

Description

Figure. Concentration-dependent activation of GRPR by GRP. Reporter cells were transfected with either the expression plasmid for gas­trin re­leas­ing pep­tide receptor (GRPR) or the mock plasmid and treated with various concentrations of gas­trin-re­leas­ing pep­tide (GRP). Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 1.3 nM.