GRPR

Figure. Concentration-dependent activation of GRPR by GRP
Reporter cells were transfected with either the expression plasmid for gastrin releasing peptide receptor (GRPR) or the mock plasmid and treated with various concentrations of GRP. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 1.3 nM.
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
Oncology, Psychiatry, Urology/Reproduction, Non-orphan GPCRs
Symbol
GRPR
Nomenclature
gastrin releasing peptide receptor
Family
Species
Human