CNR1

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
CNR1
HGNC name
cannabinoid receptor 1
Family
Cannabinoid receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=56
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Description

Figure. Concentration-dependent activation of CNR1 by Δ9-THC. Reporter cells were transfected with the expression plasmid for can­nab­i­noid receptor 1 (CNR1) and treated with various concentrations of Δ-9-tetra­hydro­can­nab­i­nol (Δ9-THC). Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 4.1 nM.