CCKAR

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
CCKAR
HGNC name
cholecystokinin A receptor
Family
Cholecystokinin receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=76
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Description

Figure. Concentration-dependent activation of CCKAR by CCK-8. Reporter cells were transfected with the expression plasmid for chole­cysto­kinin A receptor (CCKAR) and treated with various concentrations of chole­cysto­kinin 8 (CCK-8). Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 17 nM.