FFAR1

Figure. Concentration-dependent activation of FFAR1 by TAK-875
Reporter cells were transfected with either the expression plasmid for free fatty acid receptor 1 (FFAR1) or the mock plasmid and treated with various concentrations of TAK-875. Data points shown are the mean ± SEM of an experiment, and the curve is a fit to Hill equation with an EC50 of 26 nM.
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
Endocrinology/Metabolism, Non-orphan GPCRs
Symbol
FFAR1
Nomenclature
free fatty acid receptor 1
Family
Species
Human