FFAR1

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
FFAR1
HGNC name
free fatty acid receptor 1
Family
Free fatty acid receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=225
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Description

Figure. Concentration-dependent activation of FFAR1 by TAK-875. Reporter cells were transfected with either the expression plasmid for free fatty acid receptor 1 (FFAR1) or the mock plasmid and treated with various concentrations of fasiglifam (TAK-875). Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 26 nM.