Human HRH3

Figure. Concentration-dependent activation of HRH3 by histamine

Reporter cells were transfected with either the expression plasmid for human histamine receptor H3 (HRH3) or the mock plasmid and treated with various concentrations of histamine. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 190 nM.

Nomenclature
histamine receptor H3
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Psychiatry, Neurology, Cardiology, Human non-orphan GPCRs

HRH3 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors