Human LPAR1

Figure. Concentration-dependent activation of LPAR1 by LPA

Reporter cells were transfected with either the expression plasmid for human lysophosphatidic acid receptor 1 (LPAR1) or the mock plasmid and treated with various concentrations of LPA. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 400 nM.

Nomenclature
lysophosphatidic acid receptor 1
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Oncology, Gastrointestinal, Dermatology, Musculoskeletal, Urology/Reproduction, Human non-orphan GPCRs

LPAR1 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

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