Angiotensin receptors
Overview
The actions of angiotensin II (Ang II) are mediated by AT1 and AT2 receptors, which have around 30% sequence similarity. The decapeptide angiotensin I, the octapeptide angiotensin II and the heptapeptide angiotensin III are endogenous ligands. losartan, candesartan, telmisartan, etc. are clinically used AT1 receptor blockers.Excerpt from IUPHAR/BPS Guide to Pharmacology Filters Sort resultsReset ApplyFilters Sort resultsReset Apply
Species Receptor Family Assays Human AvailableAssay modes:Agonist⋅Inverse agonist⋅Antagonist⋅PAM⋅NAMPanels:Human non-orphan GPCRs⋅Immunology/Infection⋅Oncology⋅Hematology⋅Endocrinology/Metabolism⋅Ophthalmology⋅Cardiology⋅Respiratory⋅Gastrointestinal⋅Dermatology⋅Musculoskeletal⋅Urology/Reproduction⋅à la carte Mouse AvailableAssay modes:Agonist⋅Inverse agonist⋅Antagonist⋅PAM⋅NAMPanels:Mouse non-orphan GPCRs⋅à la cartePAGE TOP