Human FFAR1

Figure. Concentration-dependent activation of FFAR1 by TAK‐875

Reporter cells were transfected with either the expression plasmid for human free fatty acid receptor 1 (FFAR1) or the mock plasmid and treated with various concentrations of TAK‐875. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 26 nM.