Figure. Concentration-dependent activation of APLNR by apelin‐13

Reporter cells were transfected with either the expression plasmid for human apelin receptor (APLNR) or the mock plasmid and treated with various concentrations of apelin‐13. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 8.1 nM.

apelin receptor
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
à la carte, Cardiology, Human non-orphan GPCRs

APLNR orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

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