Human CNR1

Figure. Concentration-dependent activation of CNR1 by Δ9‐THC

Reporter cells were transfected with either the expression plasmid for human cannabinoid receptor 1 (CNR1) or the mock plasmid and treated with various concentrations of Δ9‐THC. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 4.1 nM.

cannabinoid receptor 1
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
à la carte, Immunology/Infection, Oncology, Hematology, Endocrinology/Metabolism, Psychiatry, Neurology, Ophthalmology, Cardiology, Gastrointestinal, Dermatology, Musculoskeletal, Urology/Reproduction, Human non-orphan GPCRs

CNR1 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors