GPR119

Assay services
Available
Assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
HGNC symbol
GPR119
HGNC name
G protein-coupled receptor 119
Family
Cannabinoid receptors
Species
Human
Guide to Pharmacology link
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=126

Description

Figure. Concentration-dependent activation of GPR119 by N-oleoyl­ethanol­amine. Reporter cells were transfected with either the expression plasmid for G protein-coupled receptor 119 (GPR119) or the mock plasmid and treated with various concentrations of N-oleoyl­ethanol­amine. Data points shown are the mean ± SEM of an experiment performed in triplicate, and the curve is a fit to Hill equation with an EC50 of 6.3 µM.