GPCR Catalog

With our GPCR collection of 550 non-sensory GPCRs (300 human receptors and 250 mouse receptors) in native sequences, we provide functional assay for them in a single format, regardless of the subtypes of Gα proteins coupled. Click below for details or contact us for information about GPCRs of other animal species such as rats, rabbits, dogs, and macaque monkeys.

Species

Human

Mouse

Family

5-Hydroxytryptamine receptors

Acetylcholine receptors (muscarinic)

Adenosine receptors

Adrenoceptors

Angiotensin receptors

Apelin receptor

Bile acid receptor

Bombesin receptors

BB3 receptor

GRP

NMB

Bradykinin receptors

Calcitonin receptors

Calcium-sensing receptor

Cannabinoid receptors

Chemerin receptors

Chemokine receptors

Cholecystokinin receptors

Complement peptide receptors

Corticotropin-releasing factor receptors

CRF1 receptor

CRF2 receptor

Dopamine receptors

Endothelin receptors

Formylpeptide receptors

Free fatty acid receptors

GABAB receptors

Galanin receptors

Ghrelin receptor

Glucagon receptor family

Glycoprotein hormone receptors

Gonadotrophin-releasing hormone receptors

Histamine receptors

Hydroxycarboxylic acid receptors

Kisspeptin receptor

Leukotriene receptors

Lysophospholipid (LPA) receptors

Lysophospholipid (LPS) receptors

Lysophospholipid (S1P) receptors

Melanin-concentrating hormone receptors

Melanocortin receptors

Melatonin receptors

Metabotropic glutamate receptors

Motilin receptor

Neuromedin U receptors

Neuropeptide FF/neuropeptide AF receptors

Neuropeptide S receptor

Neuropeptide W/neuropeptide B receptors

Neuropeptide Y receptors

Neurotensin receptors

Opioid receptors

Orexin receptors

Oxoglutarate receptor

P2Y receptors

Parathyroid hormone receptors

Platelet-activating factor receptor

Prokineticin receptors

Prolactin-releasing peptide receptor

Prostanoid receptors

Proteinase-activated receptors

Proton-sensing GPCRs

QRFP receptor

Relaxin family peptide receptors

Somatostatin receptors

Steroid receptors

Succinate receptor

Tachykinin receptors

Thyrotropin-releasing hormone receptors

Trace amine receptor

Urotensin receptor

VIP and PACAP receptors

Vasopressin and oxytocin receptors

Orphan GPCRs

Panel

Human non-orphan GPCRs

Human orphan GPCRs

Mouse non-orphan GPCRs

Mouse orphan GPCRs

Non-orphan GPCRs

Orphan GPCRs

Immunology/Infection

Oncology

Hematology

Endocrinology/Metabolism

Psychiatry

Neurology

Ophthalmology

Cardiology

Respiratory

Gastrointestinal

Dermatology

Musculoskeletal

Urology/Reproduction

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Species	Receptor	Family	Assays
Human	TAAR1 trace amine associated receptor 1	Trace amine receptor	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: tyramine EC50: 880 nM
Human	UTS2R urotensin 2 receptor	Urotensin receptor	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Cardiology ⋅ Dermatology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: urotensin ⅠⅠ EC50: 92 pM
Human	AVPR1A arginine vasopressin receptor 1A	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Psychiatry ⋅ Cardiology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 510 pM
Human	AVPR1B arginine vasopressin receptor 1B	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 840 pM
Human	AVPR2 arginine vasopressin receptor 2	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Endocrinology/Metabolism ⋅ Cardiology ⋅ Musculoskeletal ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 4.8 nM
Human	OXTR oxytocin receptor	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Psychiatry ⋅ Respiratory ⋅ à la carte	Reference agonist: oxytocin EC50: 1.9 nM
Human	ADCYAP1R1 ADCYAP receptor type I	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Immunology/Infection ⋅ Hematology ⋅ Psychiatry ⋅ Respiratory ⋅ à la carte	Reference agonist: PACAP EC50: 4.4 nM
Human	VIPR1 vasoactive intestinal peptide receptor 1	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Hematology ⋅ Gastrointestinal ⋅ à la carte	Reference agonist: VIP EC50: 2.7 nM
Human	VIPR2 vasoactive intestinal peptide receptor 2	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Ophthalmology ⋅ à la carte	Reference agonist: VIP EC50: 13 nM
Human	BDKRB1 bradykinin receptor B1	Bradykinin receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	BDKRB2 bradykinin receptor B2	Bradykinin receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	CCR3 C-C motif chemokine receptor 3	Chemokine receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	C5AR2 complement component 5a receptor 2	Complement peptide receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GRM3 glutamate metabotropic receptor 3	Metabotropic glutamate receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GRM7 glutamate metabotropic receptor 7	Metabotropic glutamate receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	TBXA2R thromboxane A2 receptor	Prostanoid receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GPR34 G protein-coupled receptor 34	Lysophospholipid (LPS) receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: LPS EC50: 240 nM
Human	GPR174 G protein-coupled receptor 174	Lysophospholipid (LPS) receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: LPS EC50: 22 nM
Human	GPR4 G protein-coupled receptor 4	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR65 G protein-coupled receptor 65	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR68 G protein-coupled receptor 68	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR132 G protein-coupled receptor 132	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	P2RY8 P2Y receptor family member 8	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	AGTR2 angiotensin ⅠⅠ receptor type 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPRC6A G protein-coupled receptor class C group 6 member A	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	CCRL2 C-C motif chemokine receptor like 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	ACKR3 atypical chemokine receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR1 G protein-coupled receptor 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR3 G protein-coupled receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR6 G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR12 G protein-coupled receptor 12	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR15 G protein-coupled receptor 15	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR17 G protein-coupled receptor 17	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR18 G protein-coupled receptor 18	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR19 G protein-coupled receptor 19	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR20 G protein-coupled receptor 20	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR21 G protein-coupled receptor 21	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR22 G protein-coupled receptor 22	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR25 G protein-coupled receptor 25	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR26 G protein-coupled receptor 26	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR27 G protein-coupled receptor 27	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR31 G protein-coupled receptor 31	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR32 G protein-coupled receptor 32	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR35 G protein-coupled receptor 35	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: zaprinast EC50: 2.8 µM
Human	GPR37 G protein-coupled receptor 37	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR37L1 G protein-coupled receptor 37 like 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR39 G protein-coupled receptor 39	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR45 G protein-coupled receptor 45	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR50 G protein-coupled receptor 50	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR52 G protein-coupled receptor 52	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

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