Human ADORA1

Figure. Concentration-dependent activation of ADORA1 by NECA

Reporter cells were transfected with either the expression plasmid for human adenosine A1 receptor (ADORA1) or the mock plasmid and treated with various concentrations of NECA. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 4.8 nM.

adenosine A1 receptor
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
à la carte, Neurology, Cardiology, Respiratory, Human non-orphan GPCRs

ADORA1 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

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