Human F2RL3

Figure. Concentration-dependent activation of F2RL3 by AY‐NH2

Reporter cells were transfected with either the expression plasmid for human F2R like thrombin or trypsin receptor 3 (F2RL3) or the mock plasmid and treated with various concentrations of AY‐NH2. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 2.3 µM.

F2R like thrombin or trypsin receptor 3
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
à la carte, Hematology, Gastrointestinal, Human non-orphan GPCRs

F2RL3 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors