GPCRカタログ

感覚受容体を除くGPCRをヒト 300種、マウス 250種、計550種取り揃え、共役するGαタンパク質のサブタイプに依らず単一フォーマットのアッセイで活性を評価します。 各受容体の詳細は表をクリックしてください。また、ラット、ウサギ、イヌ、カニクイザルなど他種のGPCRについてはお問い合わせください。

Species

Human

Mouse

Family

5-Hydroxytryptamine receptors

Acetylcholine receptors (muscarinic)

Adenosine receptors

Adrenoceptors

Angiotensin receptors

Apelin receptor

Bile acid receptor

Bombesin receptors

BB3 receptor

GRP

NMB

Bradykinin receptors

Calcitonin receptors

Calcium-sensing receptor

Cannabinoid receptors

Chemerin receptors

Chemokine receptors

Cholecystokinin receptors

Complement peptide receptors

Corticotropin-releasing factor receptors

CRF1 receptor

CRF2 receptor

Dopamine receptors

Endothelin receptors

Formylpeptide receptors

Free fatty acid receptors

GABAB receptors

Galanin receptors

Ghrelin receptor

Glucagon receptor family

Glycoprotein hormone receptors

Gonadotrophin-releasing hormone receptors

Histamine receptors

Hydroxycarboxylic acid receptors

Kisspeptin receptor

Leukotriene receptors

Lysophospholipid (LPA) receptors

Lysophospholipid (LPS) receptors

Lysophospholipid (S1P) receptors

Melanin-concentrating hormone receptors

Melanocortin receptors

Melatonin receptors

Metabotropic glutamate receptors

Motilin receptor

Neuromedin U receptors

Neuropeptide FF/neuropeptide AF receptors

Neuropeptide S receptor

Neuropeptide W/neuropeptide B receptors

Neuropeptide Y receptors

Neurotensin receptors

Opioid receptors

Orexin receptors

Oxoglutarate receptor

P2Y receptors

Parathyroid hormone receptors

Platelet-activating factor receptor

Prokineticin receptors

Prolactin-releasing peptide receptor

Prostanoid receptors

Proteinase-activated receptors

Proton-sensing GPCRs

QRFP receptor

Relaxin family peptide receptors

Somatostatin receptors

Steroid receptors

Succinate receptor

Tachykinin receptors

Thyrotropin-releasing hormone receptors

Trace amine receptor

Urotensin receptor

VIP and PACAP receptors

Vasopressin and oxytocin receptors

Orphan GPCRs

Panel

Human non-orphan GPCRs

Human orphan GPCRs

Mouse non-orphan GPCRs

Mouse orphan GPCRs

Non-orphan GPCRs

Orphan GPCRs

Immunology/Infection

Oncology

Hematology

Endocrinology/Metabolism

Psychiatry

Neurology

Ophthalmology

Cardiology

Respiratory

Gastrointestinal

Dermatology

Musculoskeletal

Urology/Reproduction

à la carte

Download Catalog

Filters Sort results

Reset Apply

Species	Receptor	Family	Assays
Human	GPR61 G protein-coupled receptor 61	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR62 G protein-coupled receptor 62	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR63 G protein-coupled receptor 63	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR75 G protein-coupled receptor 75	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR78 G protein-coupled receptor 78	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR82 G protein-coupled receptor 82	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR83 G protein-coupled receptor 83	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR85 G protein-coupled receptor 85	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR87 G protein-coupled receptor 87	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR88 G protein-coupled receptor 88	Orphan GPCRs	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: 2‐PCCA EC50: 1.0 µM
Human	GPR101 G protein-coupled receptor 101	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR135 G protein-coupled receptor 135	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR139 G protein-coupled receptor 139	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR141 G protein-coupled receptor 141	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR142 G protein-coupled receptor 142	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR146 G protein-coupled receptor 146	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR148 G protein-coupled receptor 148	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR149 G protein-coupled receptor 149	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR150 G protein-coupled receptor 150	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR151 G protein-coupled receptor 151	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR152 G protein-coupled receptor 152	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR153 G protein-coupled receptor 153	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR160 G protein-coupled receptor 160	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR161 G protein-coupled receptor 161	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR162 G protein-coupled receptor 162	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR171 G protein-coupled receptor 171	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR173 G protein-coupled receptor 173	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR182 G protein-coupled receptor 182	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	LGR4 leucine rich repeat containing G protein-coupled receptor 4	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	LGR5 leucine rich repeat containing G protein-coupled receptor 5	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	LGR6 leucine rich repeat containing G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MAS1 MAS1 proto-oncogene, G protein-coupled receptor	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MAS1L MAS1 proto-oncogene like, G protein-coupled receptor	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRD MAS related GPR family member D	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRE MAS related GPR family member E	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRF MAS related GPR family member F	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRG MAS related GPR family member G	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRX1 MAS related GPR family member X1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRX2 MAS related GPR family member X2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRX3 MAS related GPR family member X3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	MRGPRX4 MAS related GPR family member X4	Orphan GPCRs	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: -	Reference agonist: sodium deoxycholate EC50: 7.5 µM
Human	TAAR2 trace amine associated receptor 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	TAAR5 trace amine associated receptor 5	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	TAAR6 trace amine associated receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	TAAR8 trace amine associated receptor 8	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	TAAR9 trace amine associated receptor 9	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR143 G protein-coupled receptor 143	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR157 G protein-coupled receptor 157	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR156 G protein-coupled receptor 156	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR158 G protein-coupled receptor 158	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

1…567…12