GPCRカタログ

感覚受容体を除くGPCRをヒト 300種、マウス 250種、計550種取り揃え、共役するGαタンパク質のサブタイプに依らず単一フォーマットのアッセイで活性を評価します。 各受容体の詳細は表をクリックしてください。また、ラット、ウサギ、イヌ、カニクイザルなど他種のGPCRについてはお問い合わせください。

Species

Human

Mouse

Family

5-Hydroxytryptamine receptors

Acetylcholine receptors (muscarinic)

Adenosine receptors

Adrenoceptors

Angiotensin receptors

Apelin receptor

Bile acid receptor

Bombesin receptors

BB3 receptor

GRP

NMB

Bradykinin receptors

Calcitonin receptors

Calcium-sensing receptor

Cannabinoid receptors

Chemerin receptors

Chemokine receptors

Cholecystokinin receptors

Complement peptide receptors

Corticotropin-releasing factor receptors

CRF1 receptor

CRF2 receptor

Dopamine receptors

Endothelin receptors

Formylpeptide receptors

Free fatty acid receptors

GABAB receptors

Galanin receptors

Ghrelin receptor

Glucagon receptor family

Glycoprotein hormone receptors

Gonadotrophin-releasing hormone receptors

Histamine receptors

Hydroxycarboxylic acid receptors

Kisspeptin receptor

Leukotriene receptors

Lysophospholipid (LPA) receptors

Lysophospholipid (LPS) receptors

Lysophospholipid (S1P) receptors

Melanin-concentrating hormone receptors

Melanocortin receptors

Melatonin receptors

Metabotropic glutamate receptors

Motilin receptor

Neuromedin U receptors

Neuropeptide FF/neuropeptide AF receptors

Neuropeptide S receptor

Neuropeptide W/neuropeptide B receptors

Neuropeptide Y receptors

Neurotensin receptors

Opioid receptors

Orexin receptors

Oxoglutarate receptor

P2Y receptors

Parathyroid hormone receptors

Platelet-activating factor receptor

Prokineticin receptors

Prolactin-releasing peptide receptor

Prostanoid receptors

Proteinase-activated receptors

Proton-sensing GPCRs

QRFP receptor

Relaxin family peptide receptors

Somatostatin receptors

Steroid receptors

Succinate receptor

Tachykinin receptors

Thyrotropin-releasing hormone receptors

Trace amine receptor

Urotensin receptor

VIP and PACAP receptors

Vasopressin and oxytocin receptors

Orphan GPCRs

Panel

Human non-orphan GPCRs

Human orphan GPCRs

Mouse non-orphan GPCRs

Mouse orphan GPCRs

Non-orphan GPCRs

Orphan GPCRs

Immunology/Infection

Oncology

Hematology

Endocrinology/Metabolism

Psychiatry

Neurology

Ophthalmology

Cardiology

Respiratory

Gastrointestinal

Dermatology

Musculoskeletal

Urology/Reproduction

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Species	Receptor	Family	Assays
Human	TAAR1 trace amine associated receptor 1	Trace amine receptor	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: tyramine EC50: 880 nM
Human	UTS2R urotensin 2 receptor	Urotensin receptor	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Cardiology ⋅ Dermatology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: urotensin ⅠⅠ EC50: 92 pM
Human	AVPR1A arginine vasopressin receptor 1A	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Psychiatry ⋅ Cardiology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 510 pM
Human	AVPR1B arginine vasopressin receptor 1B	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 840 pM
Human	AVPR2 arginine vasopressin receptor 2	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Endocrinology/Metabolism ⋅ Cardiology ⋅ Musculoskeletal ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: [R]‐vasopressin EC50: 4.8 nM
Human	OXTR oxytocin receptor	Vasopressin and oxytocin receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Psychiatry ⋅ Respiratory ⋅ à la carte	Reference agonist: oxytocin EC50: 1.9 nM
Human	ADCYAP1R1 ADCYAP receptor type I	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Immunology/Infection ⋅ Hematology ⋅ Psychiatry ⋅ Respiratory ⋅ à la carte	Reference agonist: PACAP EC50: 4.4 nM
Human	VIPR1 vasoactive intestinal peptide receptor 1	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Hematology ⋅ Gastrointestinal ⋅ à la carte	Reference agonist: VIP EC50: 2.7 nM
Human	VIPR2 vasoactive intestinal peptide receptor 2	VIP and PACAP receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Ophthalmology ⋅ à la carte	Reference agonist: VIP EC50: 13 nM
Human	BDKRB1 bradykinin receptor B1	Bradykinin receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	BDKRB2 bradykinin receptor B2	Bradykinin receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	CCR3 C-C motif chemokine receptor 3	Chemokine receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	C5AR2 complement component 5a receptor 2	Complement peptide receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GRM3 glutamate metabotropic receptor 3	Metabotropic glutamate receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GRM7 glutamate metabotropic receptor 7	Metabotropic glutamate receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	TBXA2R thromboxane A2 receptor	Prostanoid receptors	Assay modes: - Panels: -	Reference agonist: EC50:
Human	GPR34 G protein-coupled receptor 34	Lysophospholipid (LPS) receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: LPS EC50: 240 nM
Human	GPR174 G protein-coupled receptor 174	Lysophospholipid (LPS) receptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ à la carte	Reference agonist: LPS EC50: 22 nM
Human	GPR4 G protein-coupled receptor 4	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR65 G protein-coupled receptor 65	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR68 G protein-coupled receptor 68	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR132 G protein-coupled receptor 132	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	P2RY8 P2Y receptor family member 8	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	AGTR2 angiotensin ⅠⅠ receptor type 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPRC6A G protein-coupled receptor class C group 6 member A	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	CCRL2 C-C motif chemokine receptor like 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	ACKR3 atypical chemokine receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR1 G protein-coupled receptor 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR3 G protein-coupled receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR6 G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR12 G protein-coupled receptor 12	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR15 G protein-coupled receptor 15	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR17 G protein-coupled receptor 17	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR18 G protein-coupled receptor 18	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR19 G protein-coupled receptor 19	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR20 G protein-coupled receptor 20	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR21 G protein-coupled receptor 21	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR22 G protein-coupled receptor 22	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR25 G protein-coupled receptor 25	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR26 G protein-coupled receptor 26	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR27 G protein-coupled receptor 27	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR31 G protein-coupled receptor 31	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR32 G protein-coupled receptor 32	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR35 G protein-coupled receptor 35	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: zaprinast EC50: 2.8 µM
Human	GPR37 G protein-coupled receptor 37	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR37L1 G protein-coupled receptor 37 like 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR39 G protein-coupled receptor 39	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR45 G protein-coupled receptor 45	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR50 G protein-coupled receptor 50	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR52 G protein-coupled receptor 52	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

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