感覚受容体を除く全ヒトGPCR 313種を取り揃え、共役するGαタンパク質のサブタイプに依らず単一フォーマットのアッセイで活性を評価します。 各受容体の詳細は表をクリックしてください。

Family
Panel
Filters Sort results
Reset Apply
Receptor
Family
Species
Assays
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
13 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
4.0 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
2.7 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
3.2 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
3.3 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
1.9 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
2.5 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
1.7 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
26 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
85 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
8.6 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
serotonin
EC50:
1.8 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
carbachol
EC50:
310 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
carbachol
EC50:
110 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
carbachol
EC50:
31 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
carbachol
EC50:
47 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
carbachol
EC50:
5.9 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
NECA
EC50:
4.8 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
NECA
EC50:
11 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
NECA
EC50:
19 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
NECA
EC50:
1.6 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
L-phenylephrine
EC50:
18 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
L-phenylephrine
EC50:
28 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
L-phenylephrine
EC50:
67 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
noradrenaline
EC50:
71 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
noradrenaline
EC50:
33 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
noradrenaline
EC50:
89 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
isoproterenol
EC50:
22 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
isoproterenol
EC50:
26 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
isoproterenol
EC50:
47 nM
Human
Available
Assay modes:
Panels:
AGTR1
Reference agonist:
angiotensin II
EC50:
920 pM
Human
Available
Assay modes:
Panels:
Reference agonist:
apelin-13
EC50:
8.1 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
TGR5 agonist
EC50:
350 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
bombesin
EC50:
2.4 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
GRP
EC50:
1.3 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
NMB
EC50:
590 pM
Human
Available
Assay modes:
Panels:
Reference agonist:
calcitonin
EC50:
2.7 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CGRP
EC50:
1.0 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
cinacalcet
EC50:
140 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
Δ9-THC
EC50:
4.1 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
Δ9-THC
EC50:
11 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
LPI
EC50:
1.2 µM
Human
Available
Assay modes:
Panels:
Reference agonist:
N-oleoylethanolamine
EC50:
6.3 µM
Human
Available
Assay modes:
Panels:
Reference agonist:
chemerin
EC50:
15 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL3
EC50:
250 pM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL2
EC50:
1.3 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL22
EC50:
20 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL4
EC50:
7.1 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL20
EC50:
3.8 nM
Human
Available
Assay modes:
Panels:
Reference agonist:
CCL21
EC50:
15 nM
1 2 7