Last updated: November 11, 2020
We have all the 313 human non-sensory GPCRs in native sequences and provide functional assay for them in a single format, regardless of the subtypes of Gα proteins coupled. Click below for details.
HGNC symbolHGNC nameFamilyAssay servicesThumbnailAgonistEC50Synonyms
HTR1A5-hydroxytryptamine receptor 1A5-Hydroxytryptamine receptorsAvailable001_HTR1A: Dose-response curve vs SerotoninSerotonin13 nMADRBRL1|5-HT1A|ADRB2RL1|serotonin receptor 1A|Gpcr18|5-hydroxytryptamine (serotonin) receptor 1A, G protein-coupled
HTR1B5-hydroxytryptamine receptor 1B5-Hydroxytryptamine receptorsAvailable002_HTR1B: Dose-response curve vs SerotoninSerotonin4.0 nM5-HT1B|5-HT1DB|HTR1D2|5-HT1B serotonin receptor|serotonin receptor 1B|5-HT1Dβ|5-hydroxytryptamine (serotonin) receptor 1B, G protein-coupled
HTR1D5-hydroxytryptamine receptor 1D5-Hydroxytryptamine receptorsAvailable003_HTR1D: Dose-response curve vs SerotoninSerotonin2.7 nM5-HT1Dα|HTRL|5-HT1D|HT1DA|serotonin receptor 1D|Gpcr14|Htr1db|5-hydroxytryptamine (serotonin) receptor 1D, G protein-coupled
HTR1E5-hydroxytryptamine receptor 1E5-Hydroxytryptamine receptorsAvailable004_HTR1E: Dose-response curve vs SerotoninSerotonin3.2 nM5-HT1Eα|5-HT1E|5-hydroxytryptamine (serotonin) receptor 1E, G protein-coupled
HTR1F5-hydroxytryptamine receptor 1F5-Hydroxytryptamine receptorsAvailable005_HTR1F: Dose-response curve vs SerotoninSerotonin3.3 nM5-HT1Eβ|5-HT6|5-HT1F|HTR1EL|serotonin receptor 1F|5-hydroxytryptamine (serotonin) receptor 1F, G protein-coupled
HTR2A5-hydroxytryptamine receptor 2A5-Hydroxytryptamine receptorsAvailable006_HTR2A: Dose-response curve vs SerotoninSerotonin1.9 nM'D' receptor|5Ht-2|serotonin 5HT-2 receptor|serotonin receptor 2A|5-hydroxytryptamine (serotonin) receptor 2A, G protein-coupled
HTR2B5-hydroxytryptamine receptor 2B5-Hydroxytryptamine receptorsAvailable007_HTR2B: Dose-response curve vs SerotoninSerotonin2.5 nM5-HT2F|5-HT2B|serotonin receptor 2B|stomach fundus serotonin receptor|5-hydroxytryptamine (serotonin) receptor 2B, G protein-coupled
HTR2C5-hydroxytryptamine receptor 2C5-Hydroxytryptamine receptorsAvailable008_HTR2C: Dose-response curve vs SerotoninSerotonin1.7 nM5-HT1C|5-HT2C|HTR1C|5-HTR2C|5-hydroxytryptamine receptor 1C|serotonin 1c receptor|serotonin receptor 2C|5-hydroxytryptamine (serotonin) receptor 2C, G protein-coupled
HTR45-hydroxytryptamine receptor 45-Hydroxytryptamine receptorsAvailable009_HTR4: Dose-response curve vs SerotoninSerotonin26 nM5-HT4|serotonin receptor 4|5-hydroxytryptamine (serotonin) receptor 4, G protein-coupled
HTR5A5-hydroxytryptamine receptor 5A5-Hydroxytryptamine receptorsAvailable010_HTR5A: Dose-response curve vs SerotoninSerotonin85 nM5-HT|5HT5-|5-HT-5A|MR22|serotonin receptor 5A|Htr5|5-hydroxytryptamine (serotonin) receptor 5A, G protein-coupled
HTR65-hydroxytryptamine receptor 65-Hydroxytryptamine receptorsAvailable011_HTR6: Dose-response curve vs SerotoninSerotonin8.6 nM5-HT6|serotonin receptor 6|ST-B17|5-hydroxytryptamine (serotonin) receptor 6, G protein-coupled
HTR75-hydroxytryptamine receptor 75-Hydroxytryptamine receptorsAvailable012_HTR7: Dose-response curve vs SerotoninSerotonin1.8 nM5-HTx|5-HT1Y|5-HT7|GPRFO|serotonin receptor 7|5-hydroxytryptamine (serotonin) receptor 7, adenylate cyclase-coupled
CHRM1cholinergic receptor muscarinic 1Acetylcholine receptors (muscarinic)Available013_CHRM1: Dose-response curve vs CarbacholCarbachol310 nMM1 muscarinic acetylcholine receptor|Chrm-1|M1R|cholinergic receptor, muscarinic 1|cholinergic receptor|cholinergic receptor, muscarinic 1, CNS
CHRM2cholinergic receptor muscarinic 2Acetylcholine receptors (muscarinic)Available014_CHRM2: Dose-response curve vs CarbacholCarbachol110 nMM2 muscarinic acetylcholine receptor|AChR M2|Chrm-2|cholinergic receptor, muscarinic 2|cholinergic receptor|cholinergic receptor, muscarinic 2, cardiac
CHRM3cholinergic receptor muscarinic 3Acetylcholine receptors (muscarinic)Available015_CHRM3: Dose-response curve vs CarbacholCarbachol31 nMHM4|Chrm-3|M3R|cholinergic receptor, muscarinic 3|cholinergic receptor|cholinergic receptor, muscarinic 3, cardiac
CHRM4cholinergic receptor muscarinic 4Acetylcholine receptors (muscarinic)Available016_CHRM4: Dose-response curve vs CarbacholCarbachol47 nMHM3|Chrm-4|cholinergic receptor, muscarinic 4|cholinergic receptor
CHRM5cholinergic receptor muscarinic 5Acetylcholine receptors (muscarinic)Available017_CHRM5: Dose-response curve vs CarbacholCarbachol5.9 nMM5R|cholinergic receptor, muscarinic 5|cholinergic receptor
ADORA1adenosine A1 receptorAdenosine receptorsAvailable018_ADORA1: Dose-response curve vs NECANECA4.8 nMRDC7|adenosine receptor A1|A1-AR|A1R
ADORA2Aadenosine A2a receptorAdenosine receptorsAvailable019_ADORA2A: Dose-response curve vs NECANECA11 nMRDC8|A2-AR|adenosine receptor A2a
ADORA2Badenosine A2b receptorAdenosine receptorsAvailable020_ADORA2B: Dose-response curve vs NECANECA19 nMadenosine receptor A2b|A2b|A2BR
ADORA3adenosine A3 receptorAdenosine receptorsAvailable021_ADORA3: Dose-response curve vs NECANECA1.6 nMAdenosine receptor A3|TGPCR1|A3AR|ARA3
ADRA1Aadrenoceptor alpha 1AAdrenoceptorsAvailable022_ADRA1A: Dose-response curve vs L-PhenylephrineL-Phenylephrine18 nMα1c1a|ADRA1C|ADRA1L1|adrenergic alpha 1c receptor|adrenergic receptor alpha 1c|alpha 1A-adrenoceptor|alpha 1A-adrenoreceptor|alpha 1C-adrenergic receptor|alpha-1A adrenergic receptor|adrenergic receptor, alpha 1a
ADRA1Badrenoceptor alpha 1BAdrenoceptorsAvailable023_ADRA1B: Dose-response curve vs L-PhenylephrineL-Phenylephrine28 nMadrenergic alpha 1B receptor|alpha 1B-adrenoceptor|alpha 1B-adrenoreceptor|alpha1B-adrenergic receptor|adrenergic receptor
ADRA1Dadrenoceptor alpha 1DAdrenoceptorsAvailable024_ADRA1D: Dose-response curve vs L-PhenylephrineL-Phenylephrine67 nMα1a/d-adrenoceptor|α1A-adrenoceptor|α1A/D|ADRA1|ADRA1A|ADRA1R|alpha 1D-adrenoceptor|Adrd1|adrenergic receptor delta1|alpha 1D-adrenoreceptor|Adra-1|alpha1D-AR|Gpcr8
ADRA2Aadrenoceptor alpha 2AAdrenoceptorsAvailable025_ADRA2A: Dose-response curve vs NoradrenalineNoradrenaline71 nMα2D|ADRA2|ADRA2R|Adrenergic alpha 2A receptor|Adra-2|Adra-2a|alpha2A|alpha2A-adrenergic receptor|alpha2A-AR|adrenergic receptor
ADRA2Badrenoceptor alpha 2BAdrenoceptorsAvailable026_ADRA2B: Dose-response curve vs NoradrenalineNoradrenaline33 nMα2-C2|ADRA2L1|ADRA2RL1|Adrenergic alpha2B- receptor class III|alpha-2B adrenergic receptor|alpha-2B adrenoreceptor|alpha-2BAR|Adra-2b|alpha2B|adrenergic receptor
ADRA2Cadrenoceptor alpha 2CAdrenoceptorsAvailable027_ADRA2C: Dose-response curve vs NoradrenalineNoradrenaline89 nMα2-C4|ADRA2L2|ADRA2RL2|Adrenergic alpha2C- receptor class I|alpha-2 adrenergic receptor subtype C4|alpha-2C adrenergic receptor|alpha-2C adrenoreceptor|Adra-2c|adrenergic receptor
ADRB1adrenoceptor beta 1AdrenoceptorsAvailable028_ADRB1: Dose-response curve vs IsoproterenolIsoproterenol22 nMADRB1R|Adrenergic receptor beta 1|B1AR|beta-1 adrenergic receptor|beta-1 adrenoreceptor|Adrb-1|beta 1-AR|adrenergic receptor
ADRB2adrenoceptor beta 2AdrenoceptorsAvailable029_ADRB2: Dose-response curve vs IsoproterenolIsoproterenol26 nMADRB2R|ADRBR|B2AR|beta-2 adrenergic receptor|beta-2 adrenoreceptor|Adrb-2|beta 2-AR|Gpcr7|adrenoceptor beta 2, surface|adrenergic receptor
ADRB3adrenoceptor beta 3AdrenoceptorsAvailable030_ADRB3: Dose-response curve vs IsoproterenolIsoproterenol47 nMatypical β-adrenoceptor|ADRB|beta-3 adrenoreceptor|Adrb-3|beta 3-AR|beta3-adrenergic receptor|adrenergic receptor
AGTR1angiotensin II receptor type 1Angiotensin receptorsAvailable031_AGTR1: Dose-response curve vs Angitensin IIAngitensin II920 pMAG2S|AT2R1|AT2R1A|HAT1R|Agtr1|angiotensin II type-1 receptor|angiotensin II type-1A receptor|angiotensin II type-1B receptor|AT3|type-1A angiotensin II receptor|type-1B angiotensin II receptor|vascular type-1 angiotensin II receptor|AT1BR|Agtr-1b|Angtr-1b|Angtr-1a|AT1AR|Type-1 angiotensin II receptor|Agtr-1a|angiotensin II receptor, type 1|angiotensin II receptor, type 1a|angiotensin II receptor, type 1b|angiotensin II receptor
APLNRapelin receptorApelin receptorAvailable033_APLNR: Dose-response curve vs Apelin-13Apelin-138.1 nMangiotensin receptor-like 1|AGTRL1|APJ|APJR|angiotensin II receptor-like 1|B78|GPCR34|G-protein coupled receptor APJ|msr/apj
GPBAR1G protein-coupled bile acid receptor 1Bile acid receptorAvailable034_GPBAR1: Dose-response curve vs TGR5 agonistTGR5 agonist350 nMBG37|hGPCR19|M-BAR|TGR5|GPCR19|GPR131|GPBAR1|G protein-coupled bile acid receptor 1|membrane-type receptor for bile acids
BRS3bombesin receptor subtype 3Bombesin receptorsAvailable035_BRS3: Dose-response curve vs BombesinBombesin2.4 nMbb3|bombesin receptor subtype-3|bombesin like receptor 3
GRPRgastrin releasing peptide receptorBombesin receptorsAvailable036_GRPR: Dose-response curve vs GRPGRP1.3 nMGRP-R|BB2|GRP-preferring bombesin receptor|Gastrin-releasing peptide receptor|gastrin-releasing peptide receptor
NMBRneuromedin B receptorBombesin receptorsAvailable037_NMBR: Dose-response curve vs NMBNMB590 pMNMB-R|BB1|neuromedin B receptor|neuromedin-B-preferring bombesin receptor
CALCRcalcitonin receptorCalcitonin receptorsAvailable040_CALCR: Dose-response curve vs CalcitoninCalcitonin2.7 nMCTRI1-|CTR2|C1A/C1B|CT-R|calcitonin receptor|CTR
CALCRLcalcitonin receptor like receptorCalcitonin receptorsAvailable041_CALCRL: Dose-response curve vs CGRPCGRP1.0 nMCLR (unofficial abbreviation in common use)|CRLR
CASRcalcium sensing receptorCalcium-sensing receptorAvailable042_CASR: Dose-response curve vs CinacalcetCinacalcet140 nMCaR|GPRC2A|extracellular calcium-sensing receptor|divalent cation-sensing receptor|calcium-sensing receptor
CNR1cannabinoid receptor 1Cannabinoid receptorsAvailable044_CNR1: Dose-response curve vs Δ9-THCΔ9-THC4.1 nMCentral cannabinoid receptor|Neuronal cannabinoid receptor|THC receptor|CB-R|Cann6|SKR6R|CB1R|Cann7
CNR2cannabinoid receptor 2Cannabinoid receptorsAvailable045_CNR2: Dose-response curve vs Δ9-THCΔ9-THC11 nMrCB2|cannabinoid receptor 2 (spleen)|CB2-R|Peripheral cannabinoid receptor|cannabinoid receptor 2 (macrophage)
GPR55G protein-coupled receptor 55Cannabinoid receptorsAvailable047_GPR55: Dose-response curve vs LPILPI1.2 µM
GPR119G protein-coupled receptor 119Cannabinoid receptorsAvailable048_GPR119: Dose-response curve vs N-OleoylethanolamineN-Oleoylethanolamine6.3 µMGPCR2|glucose-dependent insulinotropic receptor|G-protein coupled receptor 2|G protein-coupled receptor 119
CMKLR1chemerin chemokine-like receptor 1Chemerin receptorsAvailable049_CMKLR1: Dose-response curve vs ChemerinChemerin15 nMChemerin1|chemokine receptor-like 1|CMKLR1|Gpcr27|G-protein coupled receptor ChemR23|G-protein coupled receptor DEZ|resolvin E1 receptor|RVER1|tazarotene induced gene 2 receptor|TIG2 receptor
CCR1C-C motif chemokine receptor 1Chemokine receptorsAvailable051_CCR1: Dose-response curve vs CCL3CCL3250 pMCC CKR1|CKR1|MIP-1α/RANTES|MIP-1αR|CD191|CMKBR1|MIP1aR|macrophage inflammatory protein-1 alpha receptor
CCR2C-C motif chemokine receptor 2Chemokine receptorsAvailable052_CCR2: Dose-response curve vs CCL2CCL21.3 nMMCP-1 receptor|CC CKR2|CKR2|CD192|chemokine receptor CCR2|CCR2A|CCR2B|chemokine (C-C motif) receptor 2
CCR4C-C motif chemokine receptor 4Chemokine receptorsAvailable054_CCR4: Dose-response curve vs CCL22CCL2220 nMCD194|ChemR13|C-C chemokine receptor 4|CC CKR4|chemokine (C-C motif) receptor 4
CCR5C-C motif chemokine receptor 5Chemokine receptorsAvailable055_CCR5: Dose-response curve vs CCL4CCL47.1 nMCHEMR13|CC CKR5|CKR5|CD195|MIP-1 alpha receptor|chemokine (C-C motif) receptor 5 (gene/pseudogene)
CCR6C-C motif chemokine receptor 6Chemokine receptorsAvailable056_CCR6: Dose-response curve vs CCL20CCL203.8 nMCKR-L3|DCCR2|GPR-CY4|STRL22|DRY-6|GPR29|CD196
CCR7C-C motif chemokine receptor 7Chemokine receptorsAvailable057_CCR7: Dose-response curve vs CCL21CCL2115 nMEBI-1|CD197
CCR8C-C motif chemokine receptor 8Chemokine receptorsAvailable058_CCR8: Dose-response curve vs CCL1CCL16.8 nMChemR1|CKR-L1|TER1|GPR-CY6
CCR9C-C motif chemokine receptor 9Chemokine receptorsAvailable059_CCR9: Dose-response curve vs CCL25CCL2515 nMGPR 9-6|GPR28
CCR10C-C motif chemokine receptor 10Chemokine receptorsAvailable060_CCR10: Dose-response curve vs CCL27CCL2727 nMGPR-2
CXCR1C-X-C motif chemokine receptor 1Chemokine receptorsAvailable065_CXCR1: Dose-response curve vs CXCL6CXCL620 nMIL8RA|IL-8 receptor type I|CD181|CKR-1|CXC-R1|high affinity interleukin-8 receptor A|CXCR1-like|IL-8 receptor α
CXCR2C-X-C motif chemokine receptor 2Chemokine receptorsAvailable066_CXCR2: Dose-response curve vs CXCL6CXCL627 nMIL8RB|IL-8R2|KC receptor|CD182|CXC-R2|GRO/MGSA receptor|high affinity interleukin-8 receptor B|CD128|Gpcr16|chemokine (C-X-C motif) receptor 2
CXCR3C-X-C motif chemokine receptor 3Chemokine receptorsAvailable067_CXCR3: Dose-response curve vs CXCL11CXCL1129 nMGPR9|CD183|MigR|G protein-coupled receptor 9|CXC-R3|interferon-inducible protein 10 receptor|IP-10 receptor|Cxcr3|CKR-L2|chemokine (C-X-C motif) receptor 3
CXCR4C-X-C motif chemokine receptor 4Chemokine receptorsAvailable068_CXCR4: Dose-response curve vs CXCL12aCXCL12a5.4 nMfusin|LCR1|LESTR|HM89|HUMSTSR|CD184|NPY3R|NPYY3R|CXCR-4|CXC-R4|SDF-1 receptor|stromal cell-derived factor 1 receptor|Cmkar4|HSY3RR|chemokine (C-X-C motif) receptor 4
CXCR5C-X-C motif chemokine receptor 5Chemokine receptorsAvailable069_CXCR5: Dose-response curve vs CXCL13CXCL1336 nMBLR-1|MDR15|NLR|CD185|Burkitt lymphoma receptor 1|CXC-R5|neurolymphatic receptor|Gpcr6
CXCR6C-X-C motif chemokine receptor 6Chemokine receptorsAvailable070_CXCR6: Dose-response curve vs CXCL16CXCL163.9 nMBONZO|TYMSTR|CD186|STRL33|chemokine (C-X-C motif) receptor 6
XCR1X-C motif chemokine receptor 1Chemokine receptorsAvailable072_XCR1: Dose-response curve vs XCL1XCL143 nMGPR5|CCXCR1|chemokine XC receptor 1|C motif-1/lymphotactin receptor
CX3CR1C-X3-C motif chemokine receptor 1Chemokine receptorsAvailable073_CX3CR1: Dose-response curve vs CX3CL1CX3CL11.8 nMCMKBRL1|Fractalkine receptor|GPR13|V28|CCRL1|CMKDR1|Rbs11|chemokine (C-X3-C motif) receptor 1
CCKARcholecystokinin A receptorCholecystokinin receptorsAvailable074_CCKAR: Dose-response curve vs CCK-8CCK-817 nMCCK1-R|cholecystokinin receptor type A|cholecystokinin-1 receptor
CCKBRcholecystokinin B receptorCholecystokinin receptorsAvailable075_CCKBR: Dose-response curve vs CCK-8CCK-8490 pMCCK2 receptor|CCK-B receptor|cholecystokinin-2 receptor|CHOLREC|gastrin/cholecystokinin type B receptor|CCK-B/gastrin receptor
C3AR1complement C3a receptor 1Complement peptide receptorsAvailable076_C3AR1: Dose-response curve vs C3aC3a3.7 nMC3AR|C3a anaphylatoxin chemotactic receptor|C3a-R|anaphylatoxin C3a receptor|complement component 3a receptor 1
C5AR1complement C5a receptor 1Complement peptide receptorsAvailableCD88|C5A|C5AR|C5R1|C5a anaphylatoxin chemotactic receptor|C5a-R|complement C5a receptor|complement component 5a receptor 1|C5aR1
CRHR1corticotropin releasing hormone receptor 1Corticotropin-releasing factor receptorsAvailable079_CRHR1: Dose-response curve vs CRHCRH22 nMCRFR1|CRF-R|CRHR|CRH-R1|CRF-R1alpha|CRF 1 receptor|CRF-RA
CRHR2corticotropin releasing hormone receptor 2Corticotropin-releasing factor receptorsAvailable080_CRHR2: Dose-response curve vs UrocortinUrocortin23 nMCRFR2|CRF-R2|CRH-R2|CRF 2 receptor|CRFR2alpha|CRFR2beta
DRD1dopamine receptor D1Dopamine receptorsAvailable081_DRD1: Dose-response curve vs DopamineDopamine260 nMD1A|DADR|Gpcr15|dopamine D1 receptor|Dopamine-1A receptor|D1 receptor
DRD2dopamine receptor D2Dopamine receptorsAvailable082_DRD2: Dose-response curve vs DopamineDopamine260 nMD2A and D2B|dopamine D2 receptor|dopamine receptor 2|D2 receptor|D2R|D2(415) and D2(444)
DRD3dopamine receptor D3Dopamine receptorsAvailable083_DRD3: Dose-response curve vs DopamineDopamine220 nMD3 receptor|dopamine D3 receptor|dopaminergic receptor D3|D3R
DRD4dopamine receptor D4Dopamine receptorsAvailable084_DRD4: Dose-response curve vs DopamineDopamine260 nMd(2C) dopamine receptor|dopamine receptor 4|D4R
DRD5dopamine receptor D5Dopamine receptorsAvailable085_DRD5: Dose-response curve vs DopamineDopamine250 nMDRD1B|DRD1L2|D(1B) dopamine receptor|dopamine receptor 5|Gpcr1
EDNRAendothelin receptor type AEndothelin receptorsAvailable086_EDNRA: Dose-response curve vs ET-1ET-15.5 nMENDOR|endothelin A receptor|endothelin-1 receptor|ET-AR|Gpcr10
EDNRBendothelin receptor type BEndothelin receptorsAvailable087_EDNRB: Dose-response curve vs ET-1ET-15.0 nMHSCR|HSCR2|endothelin B receptor|ET-BR
GPR183G protein-coupled receptor 183Steroid receptorsAvailable089_GPR183: Dose-response curve vs 7α,25-dihydroxycholesterol7α,25-dihydroxycholesterol2.0 nMEBI2|Epstein-Barr virus-induced gene 2|EBV-induced G protein-coupled receptor 2|G protein-coupled receptor 183|lymphocyte-specific G protein-coupled receptor
FPR1formyl peptide receptor 1Formylpeptide receptorsAvailable090_FPR1: Dose-response curve vs fMLPfMLP3.5 nMNFPR|FPR|formyl peptide receptor 1|fMLF-R
FPR2formyl peptide receptor 2Formylpeptide receptorsAvailable091_FPR2: Dose-response curve vs WKYMVMWKYMVM940 pMALXR|FMLPX|FPRH1|LXA4R|ALX|FPRH2|FPRL1|RFP|formyl peptide receptor-like 1|formyl peptide receptor 2|formyl peptide receptor, related sequence 2|Fpr-rs2|ALX/FPR2|FPR2A
FPR3formyl peptide receptor 3Formylpeptide receptorsAvailable092_FPR3: Dose-response curve vs WKYMVMWKYMVM460 nMFMLPY|FPRH1|FPRL2|Fprl1|Lxa4r|LXA4-R
FFAR1free fatty acid receptor 1Free fatty acid receptorsAvailable093_FFAR1: Dose-response curve vs TAK-875TAK-87526 nMGPR40|FFA1R|G protein-coupled receptor 40
FFAR3free fatty acid receptor 3Free fatty acid receptorsAvailable094_FFAR3: Dose-response curve vs Propionate NaPropionate Na880 µMFFA3R|GPR41|LSSIG|G protein-coupled receptor 41|GPCR41
FFAR2free fatty acid receptor 2Free fatty acid receptorsAvailable095_FFAR2: Dose-response curve vs Acetic acidAcetic acid100 µMFFA2R|GPCR3|GPR43|G protein-coupled receptor 43
GPR84G protein-coupled receptor 84Free fatty acid receptorsAvailable096_GPR84: Dose-response curve vs ZQ-16ZQ-162.2 µMGPCR4|Inflammation-related G-protein coupled receptor EX33
FFAR4free fatty acid receptor 4Free fatty acid receptorsAvailable097_FFAR4: Dose-response curve vs GPR120 cpdAGPR120 cpdA1.9 µMPGR4|GPR120|GPR129|G-protein-coupled receptor GT01|GT01|G protein-coupled receptor 120|G protein-coupled receptor 129|omega-3 fatty acid receptor 1|O3FAR1|G-protein coupled receptor GT01
GABBR1gamma-aminobutyric acid type B receptor subunit 1GABAB receptorsAvailable098_GABBR1: Dose-response curve vs BaclofenBaclofen9.4 µMGABABR1|GPRC3A|GABA-B receptor 1|GABABR1|gamma-aminobutyric acid (GABA) B receptor 1|gamma-aminobutyric acid (GABA) B receptor
GABBR2gamma-aminobutyric acid type B receptor subunit 2GABAB receptorsAvailable099_GABBR2: Dose-response curve vs BaclofenBaclofen9.4 µMGABABR1|GPRC3A|GABA-B receptor 1|GABABR1|gamma-aminobutyric acid (GABA) B receptor 1|gamma-aminobutyric acid (GABA) B receptor
GALR1galanin receptor 1Galanin receptorsAvailable100_GALR1: Dose-response curve vs GalaninGalanin1.9 nMGALNR|GALNR1
GALR2galanin receptor 2Galanin receptorsAvailable101_GALR2: Dose-response curve vs GalaninGalanin1.3 nMGALNR2
GALR3galanin receptor 3Galanin receptorsGALR3|Galnr3
GHSRgrowth hormone secretagogue receptorGhrelin receptorAvailable104_GHSR: Dose-response curve vs GhrelinGhrelin4.0 nMgrowth hormone-releasing peptide receptor|GH-releasing peptide receptor|GHS-R|ghrelin receptor 1a
GHRHRgrowth hormone releasing hormone receptorGlucagon receptor familyAvailable105_GHRHR: Dose-response curve vs GHRHGHRH2.0 nMGRF receptor|GRFR|growth hormone-releasing factor receptor|Ghrfr
GIPRgastric inhibitory polypeptide receptorGlucagon receptor familyAvailable106_GIPR: Dose-response curve vs GIPGIP3.4 nMGippr|GIP-R
GLP1Rglucagon like peptide 1 receptorGlucagon receptor familyAvailable107_GLP1R: Dose-response curve vs GLP1-(7-36)amideGLP1-(7-36)amide7.6 nMGLP-1R|glucagon-like peptide 1 receptor
GLP2Rglucagon like peptide 2 receptorGlucagon receptor familyAvailable108_GLP2R: Dose-response curve vs GLP2GLP27.4 nMGLP-2R
GCGRglucagon receptorGlucagon receptor familyAvailable109_GCGR: Dose-response curve vs GlucagonGlucagon6.3 nMGGR|GL-R|GR
SCTRsecretin receptorGlucagon receptor familyAvailable110_SCTR: Dose-response curve vs SecretinSecretin7.6 nMSCT-R
FSHRfollicle stimulating hormone receptorGlycoprotein hormone receptorsAvailable111_FSHR: Dose-response curve vs FSHFSH8.6 ng/mlFollitropin receptor|LGR1|FSH-R
LHCGRluteinizing hormone/choriogonadotropin receptorGlycoprotein hormone receptorsAvailable112_LHCGR: Dose-response curve vs rLHα/βrLHα/β26 ng/mlChoriogonadotropin receptor|LCGR|LGR2|LHR|lutropin-choriogonadotropic hormone receptor|LH-R
TSHRthyroid stimulating hormone receptorGlycoprotein hormone receptorsAvailable113_TSHR: Dose-response curve vs TSHTSH18 ng/mlThyrotropin Receptor|LGR3|TSH-R
GNRHRgonadotropin releasing hormone receptorGonadotrophin-releasing hormone receptorsAvailable114_GNRHR: Dose-response curve vs LH-RHLH-RH93 pMluteinizing hormone-releasing hormone (LHRH) receptor|GNRHR1|LHRH receptor|Type I GnRHR|gnRH receptor|GnRH-R|GnRH I receptor|GnRHR|luliberin receptor|LHRHR
HRH1histamine receptor H1Histamine receptorsAvailable115_HRH1: Dose-response curve vs HistamineHistamine17 nMH1R|HH1R|Hisr
HRH2histamine receptor H2Histamine receptorsAvailable116_HRH2: Dose-response curve vs HistamineHistamine240 nMgastric receptor I|H2R|HH2R
HRH3histamine receptor H3Histamine receptorsAvailable117_HRH3: Dose-response curve vs HistamineHistamine190 nMGPCR97|H3R|HH3R
HRH4histamine receptor H4Histamine receptorsAvailable118_HRH4: Dose-response curve vs HistamineHistamine51 nMGPCR105|HH4R|H4R
HCAR1hydroxycarboxylic acid receptor 1Hydroxycarboxylic acid receptorsFKSG80|LACR1|lactate receptor 1|T-cell activation G protein-coupled receptor|G protein-coupled receptor 104|G protein-coupled receptor 81|Gpr81
HCAR2hydroxycarboxylic acid receptor 2Hydroxycarboxylic acid receptorsAvailable120_HCAR2: Dose-response curve vs Nicotinic acidNicotinic acid5.8 µMPUMAG|G-protein coupled receptor HM74A|Nicotinic acid receptor|Nic1|G protein-coupled receptor 109A|Niacr1|niacin receptor 1
HCAR3hydroxycarboxylic acid receptor 3Hydroxycarboxylic acid receptorsAvailable121_HCAR3: Dose-response curve vs 3-OH-octanoic acid3-OH-octanoic acid130 µMNIACR2|Low affinity nicotinic acid receptor|Nic2|G protein-coupled receptor 109B
KISS1RKISS1 receptorKisspeptin receptorAvailable122_KISS1R: Dose-response curve vs Kisspeptin-10Kisspeptin-101.3 nMGPR54|Metastin receptor|hOT7T175|kiSS-1 receptor|kiSS-1R|KiSS1-derived peptide receptor
LTB4Rleukotriene B4 receptorLeukotriene receptorsAvailable123_LTB4R: Dose-response curve vs LTB4LTB484 pMBLTR|GPR16
LTB4R2leukotriene B4 receptor 2Leukotriene receptorsAvailable124_LTB4R2: Dose-response curve vs LTB4LTB436 nMBLTR2|LTB4 receptor JULF2|LTB4-R2|12-HHT receptor|NOP9
CYSLTR1cysteinyl leukotriene receptor 1Leukotriene receptorsAvailable125_CYSLTR1: Dose-response curve vs LTD4LTD47.9 nMHG55|LTD4|CYSLT1R|leukotriene D4 receptor
CYSLTR2cysteinyl leukotriene receptor 2Leukotriene receptorsAvailable126_CYSLTR2: Dose-response curve vs LTD4LTD4400 pMLTC4|CYSLT2R|HG57
OXER1oxoeicosanoid receptor 1Leukotriene receptorsAvailable127_OXER1: Dose-response curve vs 5-oxo-ETE5-oxo-ETE130 nMhGPCR48|R527|TG1019|GPR170|5-oxo-ETE receptor|oxoeicosanoid (OXE) receptor 1
PTAFRplatelet activating factor receptorPlatelet-activating factor receptorAvailable128_PTAFR: Dose-response curve vs CH3-cabamyl PAF C-16CH3-cabamyl PAF C-16840 pMPAFr|AGEPC receptor
LPAR1lysophosphatidic acid receptor 1Lysophospholipid (LPA) receptorsAvailable129_LPAR1: Dose-response curve vs LPALPA400 nMEDG2|GPR26|VZG1|endothelial differentiation gene 2, lysophosphatidic acid G-protein-coupled receptor, 2|LPA receptor 1|Lpar1|lysophosphatidic acid receptor Edg-2
LPAR2lysophosphatidic acid receptor 2Lysophospholipid (LPA) receptorsAvailable130_LPAR2: Dose-response curve vs LPALPA1.7 µMEdg4|Pbx4|pre-B-cell leukemia transcription factor 4|endothelial differentiation gene 4, lysophosphatidic acid G-protein-coupled receptor 4
LPAR3lysophosphatidic acid receptor 3Lysophospholipid (LPA) receptorsAvailable131_LPAR3: Dose-response curve vs LPALPA1.3 µMEdg7|LPA receptor 3|endothelial differentiation gene 7, lysophosphatidic acid G-protein-coupled receptor 7
LPAR4lysophosphatidic acid receptor 4Lysophospholipid (LPA) receptorsAvailable132_LPAR4: Dose-response curve vs LPALPA2.1 µMP2RY9|P2Y5-like receptor|GPR23|G protein-coupled receptor 23|LPA receptor 4|LPA4|P2Y purinoceptor 9|Purinergic receptor 9
LPAR5lysophosphatidic acid receptor 5Lysophospholipid (LPA) receptorsAvailable133_LPAR5: Dose-response curve vs LPALPA3.0 µMGPR93|LPAR5|GPR92|G protein-coupled receptor 92
LPAR6lysophosphatidic acid receptor 6Lysophospholipid (LPA) receptorsAvailable134_LPAR6: Dose-response curve vs LPALPA750 nMP2RY5|LPA receptor 6|oleoyl-L-alpha-lysophosphatidic acid receptor|P2Y purinoceptor 5|purinergic receptor 5
S1PR1sphingosine-1-phosphate receptor 1Lysophospholipid (S1P) receptorsAvailable135_S1PR1: Dose-response curve vs S1PS1P7.5 nMCD363|EDG1 (Edg1)|endothelial differentiation G protein-coupled receptor 1
S1PR2sphingosine-1-phosphate receptor 2Lysophospholipid (S1P) receptorsAvailable136_S1PR2: Dose-response curve vs S1PS1P110 nMedg5|Gpcr13|endothelial differentiation G protein-coupled receptor 5|G protein-coupled receptor 13|GPCR18|S1P receptor 2
S1PR3sphingosine-1-phosphate receptor 3Lysophospholipid (S1P) receptorsAvailable137_S1PR3: Dose-response curve vs S1PS1P23 nMedg3|endothelial differentiation G protein-coupled receptor 3
S1PR4sphingosine-1-phosphate receptor 5Lysophospholipid (S1P) receptorsedg6|endothelial differentiation, G protein-coupled receptor 6
S1PR5sphingosine-1-phosphate receptor 5Lysophospholipid (S1P) receptorsAvailable139_S1PR5: Dose-response curve vs S1PS1P34 nMedg8|NRG-1|endothelial differentiation G protein-coupled receptor 8|nerve growth factor-regulated G-protein-coupled receptor 1
MCHR1melanin concentrating hormone receptor 1Melanin-concentrating hormone receptorsAvailable140_MCHR1: Dose-response curve vs MCHMCH37 nMGPR24|MCH1R|G protein-coupled receptor 24|MCH receptor 1|somatostatin receptor-like protein
MCHR2melanin concentrating hormone receptor 2Melanin-concentrating hormone receptorsAvailable141_MCHR2: Dose-response curve vs MCHMCH2.1 nMGPR145|GPRv17|MCH2R|G protein-coupled receptor 145|melanin-concentrating hormone receptor 2
MC1Rmelanocortin 1 receptorMelanocortin receptorsAvailable142_MC1R: Dose-response curve vs α-MSHα-MSH850 pMMSH-R|melanocortin 1 receptor (alpha melanocyte stimulating hormone receptor)
MC2Rmelanocortin 2 receptorMelanocortin receptorsAvailable143_MC2R: Dose-response curve vs ACTHACTH4.1 nMACTHR|melanocortin 2 receptor|adrenocorticotropic hormone receptor|melanocortin 2 receptor (adrenocorticotropic hormone)
MC3Rmelanocortin 3 receptorMelanocortin receptorsAvailable144_MC3R: Dose-response curve vs α-MSHα-MSH180 pMγ-MSH receptor|melanocortin receptor 3
MC4Rmelanocortin 4 receptorMelanocortin receptorsAvailable145_MC4R: Dose-response curve vs α-MSHα-MSH600 pM
MC5Rmelanocortin 5 receptorMelanocortin receptorsAvailable146_MC5R: Dose-response curve vs α-MSHα-MSH8.5 nMMC5R|melanocortin receptor 5
MTNR1Amelatonin receptor 1AMelatonin receptorsAvailable147_MTNR1A: Dose-response curve vs MelatoninMelatonin100 pMmel1a receptor|MelR
MTNR1Bmelatonin receptor 1BMelatonin receptorsAvailable148_MTNR1B: Dose-response curve vs MelatoninMelatonin95 pMmel1b receptor
GRM1glutamate metabotropic receptor 1Metabotropic glutamate receptorsAvailable149_GRM1: Dose-response curve vs L-Glutamic acidL-Glutamic acid6.4 µMGPRC1A|metabotropic glutamate receptor 1|wobl|MGLUR1|SCAR13|glutamate receptor, metabotropic 1|glutamate receptor
GRM2glutamate metabotropic receptor 2Metabotropic glutamate receptorsAvailable150_GRM2: Dose-response curve vs L-Glutamic acidL-Glutamic acid6.4 µMmGluR2|GPRC1B|metabotropic glutamate receptor 2|glutamate receptor
GRM4glutamate metabotropic receptor 4Metabotropic glutamate receptorsAvailable152_GRM4: Dose-response curve vs L-Glutamic acidL-Glutamic acid34 µMmGluR4|GPRC1D|glutamate receptor
GRM5glutamate metabotropic receptor 5Metabotropic glutamate receptorsAvailable153_GRM5: Dose-response curve vs L-Glutamic acidL-Glutamic acid5.9 µMmGluR5|GPRC1E|glutamate receptor
GRM6glutamate metabotropic receptor 6Metabotropic glutamate receptorsAvailable154_GRM6: Dose-response curve vs L-Glutamic acidL-Glutamic acid190 µMGprc1f|mGluR6|nob4|nerg1|nob2|nob3|glutamate receptor
GRM8glutamate metabotropic receptor 8Metabotropic glutamate receptorsAvailable156_GRM8: Dose-response curve vs L-Glutamic acidL-Glutamic acid26 µMGprc1h|mGluR8|GLUR8|mGluR8b|glutamate receptor
MLNRmotilin receptorMotilin receptorAvailable157_MLNR: Dose-response curve vs MotilinMotilin590 pMMOT-R|MTLR|GPR38|MTLR1|G protein-coupled receptor 38
NMUR1neuromedin U receptor 1Neuromedin U receptorsAvailable158_NMUR1: Dose-response curve vs MNU-23MNU-231.3 nMGPR66|FM-3|NmU-R1|SNORF62
NMUR2neuromedin U receptor 2Neuromedin U receptorsAvailable159_NMUR2: Dose-response curve vs MNU-23MNU-23390 pMFM-4|FM4|SNORF72|NMU-R2|TGR-1
NPFFR1neuropeptide FF receptor 1Neuropeptide FF/neuropeptide AF receptorsAvailable160_NPFFR1: Dose-response curve vs NPFFNPFF22 nMGPR147|G protein-coupled receptor 147|NPFF1|RFamide-related peptide receptor OT7T022|NPFF1R1|OT7T022|GnIH-R|GnIH-R/RFRP-3
NPFFR2neuropeptide FF receptor 2Neuropeptide FF/neuropeptide AF receptorsAvailable161_NPFFR2: Dose-response curve vs NPFFNPFF280 pMF8Famide receptor|GPR74|NPGPR|G protein-coupled receptor 74
NPSR1neuropeptide S receptor 1Neuropeptide S receptorAvailable162_NPSR1: Dose-response curve vs NPSNPS260 nMVRR1|GPR154|PGR14|G protein-coupled receptor 154|vasopressin receptor-related receptor 1
NPBWR1neuropeptides B and W receptor 1Neuropeptide W/neuropeptide B receptorsAvailable163_NPBWR1: Dose-response curve vs NPW-30NPW-3020 nMGPR7|G protein-coupled receptor 7|neuropeptides B/W receptor type 1
NPBWR2neuropeptides B and W receptor 2Neuropeptide W/neuropeptide B receptorsAvailable164_NPBWR2: Dose-response curve vs NPW-30NPW-3014 nMGPR8|G protein-coupled receptor 8|neuropeptides B/W receptor 2
NPY1Rneuropeptide Y receptor Y1Neuropeptide Y receptorsAvailable165_NPY1R: Dose-response curve vs NPYNPY840 pMNPY-Y1 receptor|FC5|neuropeptide Y receptor type 1|Y1-R
NPY2Rneuropeptide Y receptor Y2Neuropeptide Y receptorsAvailable166_NPY2R: Dose-response curve vs NPYNPY4.6 nMneuropeptide Y receptor type 2|NPY-Y2 receptor
NPY4Rneuropeptide Y receptor Y4Neuropeptide Y receptorsAvailable167_NPY4R: Dose-response curve vs NPYNPY29 nMPP1|neuropeptide Y receptor type 4|pancreatic polypeptide receptor 1
NPY5Rneuropeptide Y receptor Y5Neuropeptide Y receptorsAvailable168_NPY5R: Dose-response curve vs NPYNPY7.6 nMfood intake receptor|neuropeptide Y receptor type 5
NTSR1neurotensin receptor 1Neurotensin receptorsAvailable169_NTSR1: Dose-response curve vs NeurotensinNeurotensin180 pMNTR1|NTRH|NTSR1|NTR|neurotensin receptor type 1|Levocabastin-insensitive neurotensin receptor|NT-1R|neurotensin receptor 1 (high affinity)
NTSR2neurotensin receptor 2Neurotensin receptorsAvailable170_NTSR2: Dose-response curve vs SR48692SR4869283 nMlevocabastine-sensitive neurotensin receptor|NTRL|NTR2|high-affinity levocabastine-sensitive neurotensin receptor|neurotensin receptor type 2|NT2R
OPRD1opioid receptor delta 1Opioid receptorsAvailable171_OPRD1: Dose-response curve vs Leu-enkephalinLeu-enkephalin6.1 nMDOP|DOR|OP1|Delta receptor|DOR-1|DOPr|opioid receptor
OPRK1opioid receptor kappa 1Opioid receptorsAvailable172_OPRK1: Dose-response curve vs Dynorphin ADynorphin A8.2 nMKOR-1|Kappa receptor|OP2|KOP|KOPr
OPRM1opioid receptor mu 1Opioid receptorsAvailable173_OPRM1: Dose-response curve vs DAMGODAMGO21 nMMu receptor|MOP|OP3|MOPr|opioid receptor, mu 1|opioid receptor
OPRL1opioid related nociceptin receptor 1Opioid receptorsAvailable174_OPRL1: Dose-response curve vs NociceptinNociceptin290 pMN/OFQ receptor|OP4|KOR-3|NOCIR|kappa3-related opioid receptor|MOR-C|nociceptin receptor ORL1|XOR1|NOP-r|nociceptin/orphanin FQ receptor|NOPr
HCRTR1hypocretin receptor 1Orexin receptorsAvailable175_HCRTR1: Dose-response curve vs Orexin AOrexin A1.6 nMOX1R|Hctr1|hypocretin receptor 1|orexin receptor type 1|hypocretin (orexin) receptor 1
HCRTR2hypocretin receptor 2Orexin receptorsAvailable176_HCRTR2: Dose-response curve vs Orexin AOrexin A3.0 nMhypocretin receptor 2|orexin receptor type 2|OX2R|hypocretin (orexin) receptor 2
OXGR1oxoglutarate receptor 1Oxoglutarate receptorsAvailable177_OXGR1: Dose-response curve vs 2-Oxoglutaric acid2-Oxoglutaric acid66 µMP2RY15|GPR80|GPR99|P2Y15|2-oxoglutarate receptor 1|Alpha-ketoglutarate receptor 1|G protein-coupled receptor 99|P2Y purinoceptor 15|G protein-coupled receptor 80
P2RY1purinergic receptor P2Y1P2Y receptorsAvailable178_P2RY1_ADP: Dose-response curve vs ADPADP3.3 µMATP receptor|P2 purinoceptor subtype Y1|P2Y purinoceptor 1|platelet ADP receptor|Purinergic receptor P2Y1|P2Y ATP receptor 1|P2Y1 receptor|purinergic receptor P2Y
P2RY2purinergic receptor P2Y2P2Y receptorsAvailable179_P2RY2_UTP: Dose-response curve vs UTPUTP1.5 µMATP receptor|P2U purinoceptor 1|P2Y ATP receptor 2|P2Y purinoceptor 2|purinergic receptor P2Y
P2RY4pyrimidinergic receptor P2Y4P2Y receptorsAvailable180_P2RY4_ATP: Dose-response curve vs ATPATP27 µMpyrimidinoceptor|uridine nucleotide receptor|NRU|UNR|P2Y ATP receptor 4|P2Y purinoceptor 4|P2Y4R|pyrimidinergic receptor P2Y
P2RY6pyrimidinergic receptor P2Y6P2Y receptorsAvailable181_P2RY6_UDP: Dose-response curve vs UDPUDP96 nMuridine nucleotide receptor|P2Y6|P2Y ATP receptor 6|P2Y purinoceptor 6|pyrimidinergic receptor P2Y
P2RY11purinergic receptor P2Y11P2Y receptorsAvailable182_P2RY11_ATP: Dose-response curve vs ATPATP13 µMpurinergic receptor P2Y, G-protein coupled, 11
P2RY12purinergic receptor P2Y12P2Y receptorsAvailable183_P2RY12_ADP: Dose-response curve vs ADPADP3.0 µMSP1999|P2YADP|HORK3|P2Y purinoceptor 12|P2Y12 platelet ADP receptor|purinergic receptor P2Y
P2RY13purinergic receptor P2Y13P2Y receptorsGPR94|G protein-coupled receptor 86|P2Y purinoceptor 13|purinergic receptor P2Y, G-protein coupled 13|purinergic receptor P2Y
P2RY14purinergic receptor P2Y14P2Y receptorsAvailable185_P2RY14_UDP-glucose: Dose-response curve vs UDP-glucoseUDP-glucose160 nMG protein coupled receptor for UDP-glucose|G protein-coupled receptor 105|GPR105|P2Y purinoceptor 14|G-protein coupled receptor 105|purinergic receptor P2Y
P2RY8P2Y receptor family member 8Orphan receptorsAvailableG-protein coupled purinergic receptor P2Y8|P2Y purinoceptor 8|purinergic receptor P2Y8
P2RY10P2Y receptor family member 10P2Y receptorsAvailable187_P2RY10_LPS: Dose-response curve vs LPSLPS310 nMpurinergic receptor P2Y10|purinergic receptor P2Y, G-protein coupled 10|purinergic receptor P2Y
PTH1Rparathyroid hormone 1 receptorParathyroid hormone receptorsAvailable188_PTH1R: Dose-response curve vs PTHPTH2.2 nMPPR|PTHR|PTHR1
PTH2Rparathyroid hormone 2 receptorParathyroid hormone receptorsAvailable189_PTH2R: Dose-response curve vs PTHPTH9.0 nMPTHR2
PROKR1prokineticin receptor 1Prokineticin receptorsAvailable190_PROKR1: Dose-response curve vs Prokineticin2Prokineticin215 ng/mlGPR73a|VEGFR-1|ZAQ|GPR73|G-protein coupled receptor ZAQ|G protein-coupled receptor 73
PROKR2prokineticin receptor 2Prokineticin receptorsAvailable191_PROKR2: Dose-response curve vs Prokineticin2Prokineticin225 ng/mlGPR73b|VEGFR-2|GPR73a|GPRg2|I5E
PRLHRprolactin releasing hormone receptorProlactin-releasing peptide receptorAvailable192_PRLHR: Dose-response curve vs PrRp-31PrRp-311.8 nMPrRPR|GPR10|G protein-coupled receptor 10|prRP receptor
PTGDRprostaglandin D2 receptorProstanoid receptorsAvailable193_PTGDR: Dose-response curve vs BW245CBW245C380 pMDP1|prostanoid DP receptor-like|PTGDR1|prostaglandin D2 receptor (DP)
PTGDR2prostaglandin D2 receptor 2Prostanoid receptorsAvailable194_PTGDR2: Dose-response curve vs (15)-15-CH3-PGD2(15)-15-CH3-PGD26.8 nMCRTH2|CD294|G protein-coupled receptor 44|prostaglandin D2 receptor 2|PGD2 receptor|Gpr44
PTGER1prostaglandin E receptor 1Prostanoid receptorsAvailable195_PTGER1: Dose-response curve vs SulprostoneSulprostone26 nMEP1 prostanoid receptor|PGE receptor EP1 subtype|prostanoid EP1 receptor|prostaglandin E receptor 1 (subtype EP1), 42kDa
PTGER2prostaglandin E receptor 2Prostanoid receptorsAvailable196_PTGER2: Dose-response curve vs MisoprostolMisoprostol62 nMPGE receptor EP2 subtype|prostanoid EP2 receptor|Ptger-ep2|prostaglandin E receptor 2 (subtype EP2), 53kDa
PTGER3prostaglandin E receptor 3Prostanoid receptorsAvailable197_PTGER3: Dose-response curve vs MisoprostolMisoprostolPGE receptor EP3 subtype|prostaglandin E receptor 3|prostanoid EP3 receptor
PTGER4prostaglandin E receptor 4Prostanoid receptorsAvailable198_PTGER4: Dose-response curve vs MisoprostolMisoprostol840 nMEP2|PGE receptor EP4 subtype|prostanoid EP4 receptor
PTGFRprostaglandin F receptorProstanoid receptorsAvailable199_PTGFR: Dose-response curve vs FluprostenolFluprostenol98 pMPF2AR|PGF receptor|PGF2 alpha receptor|prostaglandin F receptor|prostaglandin F2-alpha receptor|prostaglandin F receptor (FP)
PTGIRprostaglandin I2 receptorProstanoid receptorsAvailable200_PTGIR: Dose-response curve vs BeraprostBeraprost130 nMprostanoid IP receptor|prostacyclin receptor|prostaglandin I2 receptor|prostaglandin I2 (prostacyclin) receptor (IP)
F2Rcoagulation factor II thrombin receptorProteinase-activated receptorsAvailable202_F2R: Dose-response curve vs TFLLR-NH2TFLLR-NH2180 nMprotease-activated receptor 1|coagulation factor II (thrombin) receptor
F2RL1F2R like trypsin receptor 1Proteinase-activated receptorsAvailable203_F2RL1: Dose-response curve vs SLIGKV-NH2SLIGKV-NH2170 nMGPR11|coagulation factor II receptor-like 1|Protease-activated receptor-2|coagulation factor II (thrombin) receptor-like 1
F2RL2coagulation factor II thrombin receptor like 2Proteinase-activated receptorsAvailable204_F2RL2: Dose-response curve vs PAR-3PAR-39.2 µMcoagulation factor II receptor-like 2|protease-activated receptor 3|thrombin receptor-like 2|coagulation factor II (thrombin) receptor-like 2
F2RL3F2R like thrombin or trypsin receptor 3Proteinase-activated receptorsAvailable205_F2RL3: Dose-response curve vs AY-NH2AY-NH22.3 µMcoagulation factor II receptor-like 3|protease-activated receptor 4|thrombin receptor-like 3|coagulation factor II (thrombin) receptor-like 3|F2R like thrombin/trypsin receptor 3
QRFPRpyroglutamylated RFamide peptide receptorQRFP receptorAvailable206_QRFPR: Dose-response curve vs QRFPQRFP720 pMAQ27|SP9155|GPR103|G protein-coupled receptor 103|peptide p518 receptor
RXFP1relaxin family peptide receptor 1Relaxin family peptide receptorsAvailable207_RXFP1: Dose-response curve vs Relaxin-1Relaxin-110 nMLGR7|RXFPR1|relaxin receptor 1|leucine-rich repeat-containing G-protein-coupled receptor 7|RX1|relaxin/insulin like family peptide receptor 1
RXFP2relaxin family peptide receptor 2Relaxin family peptide receptorsAvailable208_RXFP2: Dose-response curve vs INSL3INSL3790 pMGPR106|RXFPR2|relaxin receptor 2|INSL3 receptor|leucine-rich repeat-containing G protein-coupled receptor 8|LGR8|relaxin/insulin like family peptide receptor 2
RXFP3relaxin family peptide receptor 3Relaxin family peptide receptorsAvailable209_RXFP3: Dose-response curve vs Relaxin-3Relaxin-312 nMRLN3R1|RXFPR3|GPCR135|relaxin/insulin like family peptide receptor 3
RXFP4relaxin family peptide/INSL5 receptor 4Relaxin family peptide receptorsAvailable210_RXFP4: Dose-response curve vs Relaxin-3Relaxin-329 nMRLN3R2|GPCR142|INSL5 receptor|RXFPR4|G protein-coupled receptor 100|relaxin/insulin-like family peptide receptor 4|relaxin/insulin like family peptide receptor 4
SSTR1somatostatin receptor 1Somatostatin receptorsAvailable211_SSTR1: Dose-response curve vs Somatostatin-14Somatostatin-1423 nMSRIF-2|SS1R
SSTR2somatostatin receptor 2Somatostatin receptorsAvailable212_SSTR2: Dose-response curve vs Somatostatin-14Somatostatin-143.1 nMsomatotropin release-inhibiting factor receptor|SRIF-1
SSTR3somatostatin receptor 3Somatostatin receptorsAvailable213_SSTR3: Dose-response curve vs Somatostatin-14Somatostatin-143.2 nMSRIF1C|somatostatin receptor 28|SSR-28
SSTR4somatostatin receptor 4Somatostatin receptorsAvailable214_SSTR4: Dose-response curve vs Somatostatin-14Somatostatin-14290 pMSRIF2B
SSTR5somatostatin receptor 5Somatostatin receptorsAvailable215_SSTR5: Dose-response curve vs Somatostatin-14Somatostatin-141.7 nMSOMATO
SUCNR1succinate receptor 1Succinate receptorAvailable216_SUCNR1: Dose-response curve vs Succnic acidSuccnic acid14 µMsuccinate receptor 1|GPR91|P2Y purinoceptor 1|SUCNR1|G protein-coupled receptor 91
TACR1tachykinin receptor 1Tachykinin receptorsAvailable217_TACR1: Dose-response curve vs Neurokinin ANeurokinin A990 pMSPR|Substance P receptor|NK1R|TAC1R|neurokinin receptor 1|NK1 receptor
TACR2tachykinin receptor 2Tachykinin receptorsAvailable218_TACR2: Dose-response curve vs Neurokinin ANeurokinin A570 pMNeurokinin B receptor|NKNAR|SKR|TAC2R|neurokinin A receptor|NK-2 receptor|SP-E receptor|Substance K receptor
TACR3tachykinin receptor 3Tachykinin receptorsAvailable219_TACR3: Dose-response curve vs Neurokinin ANeurokinin A27 nMNeurokinin B receptor|neurokinin beta receptor|Nmkr|Tac3r|neuromedin K receptor|NK-3 receptor|SP-N receptor
TRHRthyrotropin releasing hormone receptorThyrotropin-releasing hormone receptorsAvailable220_TRHR: Dose-response curve vs TRHTRH160 pMTRH receptor|thyroliberin receptor|TRH-R|TRH-R1
TAAR1trace amine associated receptor 1Trace amine receptorAvailable221_TAAR1: Dose-response curve vs TyramineTyramine880 nMTAR1|TaR-1|trace amine receptor 1|TRAR1
UTS2Rurotensin 2 receptorUrotensin receptorAvailable227_UTS2R: Dose-response curve vs Urotensin IIUrotensin II92 pMGPR14|UII-R1|UTR2|G protein-coupled receptor 14|urotensin II receptor|SENR (sensory epithelial neuropeptide-like receptor)
AVPR1Aarginine vasopressin receptor 1AVasopressin and oxytocin receptorsAvailable228_AVPR1A: Dose-response curve vs [R]-Vasopressin[R]-Vasopressin510 pMV1aR|AVPR1|antidiuretic hormone receptor 1a|AVPR
AVPR1Barginine vasopressin receptor 1BVasopressin and oxytocin receptorsAvailable229_AVPR1B: Dose-response curve vs [R]-Vasopressin[R]-Vasopressin840 pMAntidiuretic hormone receptor 1b|AVPR3|V3|V1bR|Vasopressin V3 receptor|VPR3|vasopressin V1b receptor|V3/V1b pituitary vasopressin receptor
AVPR2arginine vasopressin receptor 2Vasopressin and oxytocin receptorsAvailable230_AVPR2: Dose-response curve vs [R]-Vasopressin[R]-Vasopressin4.8 nMADHR|DIR3|antidiuretic hormone receptor|renal-type arginine vasopressin receptor
OXTRoxytocin receptorVasopressin and oxytocin receptorsAvailable231_OXTR: Dose-response curve vs OxtocinOxtocin1.9 nMOTR
ADCYAP1R1ADCYAP receptor type IVIP and PACAP receptorsAvailable232_ADCYAP1R1: Dose-response curve vs PACAPPACAP4.4 nMPAC1R|PVR1|PACAP receptor 1|PACAP type IA receptor|PACAPR1|pituitary adenylate cyclase activating polypeptide 1 receptor (1)|PACAP1-R|adenylate cyclase activating polypeptide 1 receptor 1|adenylate cyclase activating polypeptide 1 receptor type 1|ADCYAP receptor type 1
VIPR1vasoactive intestinal peptide receptor 1VIP and PACAP receptorsAvailable233_VIPR1: Dose-response curve vs VIPVIP2.7 nMPVR2|HVR1|RDC1|VIP and PACAP receptor 1|PACAP-R2|pituitary adenylate cyclase-activating polypeptide type II receptor|VIP-R1
VIPR2vasoactive intestinal peptide receptor 2VIP and PACAP receptorsAvailable234_VIPR2: Dose-response curve vs VIPVIP13 nMPVR3|VIP and PACAP receptor 2|PACAP-R3|pituitary adenylate cyclase-activating polypeptide type III receptor
BDKRB1bradykinin receptor B1Bradykinin receptorsB1BKR|BKR1|B1R|kinin B1 receptor|bradykinin receptor
BDKRB2bradykinin receptor B2Bradykinin receptorsB2BKR|B2BRA|BK-2 receptor|BK2R|bradykinin receptor
CCR3C-C motif chemokine receptor 3Chemokine receptorsCC CKR3|MIP-1αRL-2 (mouse)|CKR3|CC-CKR-3|CD193|chemokine (C-C motif) receptor 3
C5AR2complement component 5a receptor 2Complement peptide receptorsC5L2|C5A receptor beta|complement 5A receptor beta|G protein-coupled receptor 77|GPR77
GRM3glutamate metabotropic receptor 3Metabotropic glutamate receptorsmGluR3|GPRC1C|glutamate receptor
GRM7glutamate metabotropic receptor 7Metabotropic glutamate receptorsmGluR7|GLUR7|GPRC1G|mGlu7a receptor|glutamate receptor
TBXA2Rthromboxane A2 receptorProstanoid receptorsprostanoid TP receptor|TXA2-R
AGTR2angiotensin II receptor type 2Orphan receptorsAvailableMRX88|angiotensin receptor 2|angiotensin II type 2 receptor|AT2R|AT2-R|AT2 receptor|Agtr2|angiotensin II receptor, type 2|angiotensin II receptor
GPRC6AG protein-coupled receptor class C group 6 member AOrphan receptorsAvailableGPCR6A|G protein-coupled receptor, family C, group 6, member A|G protein-coupled receptor, class C, group 6, member A|G protein-coupled receptor
CCRL2C-C motif chemokine receptor like 2Orphan receptorsAvailableCCR11|CKRX|CRAM-A|CRAM-B|ACR5|CCR6|Chemokine receptor X
ACKR3atypical chemokine receptor 3Orphan receptorsAvailablechemokine (C-X-C motif) receptor 7|chemokine orphan receptor 1|CXCR7|Cxcr7|GPR159|G-protein coupled receptor 159|G-protein coupled receptor RDC1 homolog|RDC-1
GPR1G protein-coupled receptor 1Orphan receptorsAvailableGPR1|G protein-coupled receptor 1|Chemerin2
GPR3G protein-coupled receptor 3Orphan receptorsAvailableGpcr21|GPCR3|ACCA orphan receptor|adenylate cyclase constitutive activator|G protein-coupled receptor R4|Gpcr20
GPR4G protein-coupled receptor 4Orphan receptorsAvailableGPR19|G-protein coupled receptor 19
GPR6G protein-coupled receptor 6Orphan receptorsAvailableSphingosine 1-phosphate receptor GPR6
GPR12G protein-coupled receptor 12Orphan receptorsAvailableGpcr01|Gpcr20|GPCR21|GPCR12|R334
GPR15G protein-coupled receptor 15Orphan receptorsAvailableBOB|Brother of Bonzo
GPR17G protein-coupled receptor 17Orphan receptorsAvailableP2Y-like receptor|UDP/CysLT receptor|R12|uracil nucleotide/cysteinyl leukotriene receptor
GPR18G protein-coupled receptor 18Orphan receptorsAvailableGPCRW|NAGly receptor|N-arachidonoyol glycine receptor
GPR19G protein-coupled receptor 19Orphan receptorsAvailableGPR-NGA
GPR20G protein-coupled receptor 20Orphan receptorsAvailableGpcr5-1|P2Y4|G protein-coupled receptor 5-1
GPR21G protein-coupled receptor 21Orphan receptorsAvailable
GPR22G protein-coupled receptor 22Orphan receptorsAvailable
GPR25G protein-coupled receptor 25Orphan receptorsAvailable
GPR26G protein-coupled receptor 26Orphan receptorsAvailable
GPR27G protein-coupled receptor 27Orphan receptorsAvailablesuper conserved receptor expressed in brain 1|SREB1
GPR31G protein-coupled receptor 31Orphan receptorsAvailable12-HETER|HETER1|hydroxyeicosatetraenoic (HETE) acid receptor 1|12-(S)-HETE acid receptor|G protein-coupled receptor 31, D17Leh66c region
GPR32G protein-coupled receptor 32Orphan receptorsAvailableRvD1|RVDR1|resolvin D1 receptor
GPR34G protein-coupled receptor 34Orphan receptorsAvailable253_GPR34: Dose-response curve vs LPSLPS240 nM
GPR35G protein-coupled receptor 35Orphan receptorsAvailableG-protein coupled receptor 3|KYNA receptor|Kynurenic acid receptor
GPR37G protein-coupled receptor 37Orphan receptorsAvailableEDNRBL|EDNRLB|PAELR|hET(B)R-LP|G-protein coupled receptor CNS1|parkin-associated endothelin B-like receptor|Endothelin B receptor-like protein 1
GPR37L1G protein-coupled receptor 37 like 1Orphan receptorsAvailableCAG-18|endothelin B receptor-like protein 2|ETBRLP2|G-protein coupled receptor CNS2
GPR39G protein-coupled receptor 39Orphan receptorsAvailable
GPR45G protein-coupled receptor 45Orphan receptorsAvailablePSP24|high-affinity lysophosphatidic acid receptor|PSP24alpha|PSP24A
GPR50G protein-coupled receptor 50Orphan receptorsAvailableMTNRL|H9|Mel1c|melatonin-related receptor
GPR52G protein-coupled receptor 52Orphan receptorsAvailable
GPR61G protein-coupled receptor 61Orphan receptorsAvailableGPCR3|BALGR|biogenic amine receptor-like GPCR
GPR62G protein-coupled receptor 62Orphan receptorsAvailableGPCR8
GPR63G protein-coupled receptor 63Orphan receptorsAvailablePSP24-2|PSP24B|PSP24beta
GPR65G protein-coupled receptor 65Orphan receptorsAvailableDig1|Gpcr25|Psychosine receptor|TDAG8|T cell death associated protein 8
GPR68G protein-coupled receptor 68Orphan receptorsAvailableGPR12A|Ovarian cancer G-protein coupled receptor 1|sphingosylphosphorylcholine receptor|OGR1
GPR75G protein-coupled receptor 75Orphan receptorsAvailableWI-31133|WI31133
GPR78G protein-coupled receptor 78Orphan receptorsAvailable
GPR82G protein-coupled receptor 82Orphan receptorsAvailable
GPR83G protein-coupled receptor 83Orphan receptorsAvailableGIR|GPR72|glucocorticoid induced receptor|G protein-coupled receptor 72|JP05
GPR85G protein-coupled receptor 85Orphan receptorsAvailableSrep2|SREB2|SREB|Super conserved receptor expressed in brain 2|PKrCx1
GPR87G protein-coupled receptor 87Orphan receptorsAvailableFKSG78|GPR95
GPR88G protein-coupled receptor 88Orphan receptorsAvailableSTRG|striatum-specific G-protein coupled receptor
GPR101G protein-coupled receptor 101Orphan receptorsAvailableGPCR6
GPR132G protein-coupled receptor 132Orphan receptorsAvailableG protein-coupled receptor G2A|G2 accumulation protein
GPR135G protein-coupled receptor 135Orphan receptorsAvailableHUMNPIIY20|PAFR
GPR139G protein-coupled receptor 139Orphan receptorsAvailableG(q)-coupled orphan receptor GPRg1|GPRG1|G-protein-coupled receptor PGR3
GPR141G protein-coupled receptor 141Orphan receptorsAvailableaxor115|G-protein coupled receptor PGR13
GPR142G protein-coupled receptor 142Orphan receptorsAvailableKIF19|AXOR103|G-protein coupled receptor PGR2
GPR146G protein-coupled receptor 146Orphan receptorsAvailableAXOR120|G-protein coupled receptor PGR8
GPR148G protein-coupled receptor 148Orphan receptorsAvailableBTR|PGR6|brain and testis restricted GPCR
GPR149G protein-coupled receptor 149Orphan receptorsAvailableIEDA|G-protein coupled receptor PGR10|induced early in differentiating astrocytes gene protein
GPR150G protein-coupled receptor 150Orphan receptorsAvailablePGR11
GPR151G protein-coupled receptor 151Orphan receptorsAvailableGALR4|G-protein coupled receptor PGR7|galanin receptor 4
GPR152G protein-coupled receptor 152Orphan receptorsAvailablePGR1|PGR5|G-protein coupled receptor PGR5
GPR153G protein-coupled receptor 153Orphan receptorsAvailablePGR1
GPR160G protein-coupled receptor 160Orphan receptorsAvailableGPCR1|GPCR150
GPR161G protein-coupled receptor 161Orphan receptorsAvailableG-protein coupled receptor RE2
GPR162G protein-coupled receptor 162Orphan receptorsAvailableGRCA
GPR171G protein-coupled receptor 171Orphan receptorsAvailableG-protein coupled receptor H963|platelet activating receptor homolog
GPR173G protein-coupled receptor 173Orphan receptorsAvailableSREB3|Super conserved receptor expressed in brain 3
GPR174G protein-coupled receptor 174Orphan receptorsAvailable287_GPR174: Dose-response curve vs LPSLPS22 nMFKSG79
GPR182G protein-coupled receptor 182Orphan receptorsAvailableADMR|Gpcr22|NOW|adrenomedullin receptor|L1-R|Gpcr17
LGR4leucine rich repeat containing G protein-coupled receptor 4Orphan receptorsAvailableGPR48|leucine-rich repeat-containing G protein-coupled receptor 4|leucine-rich repeat containing G protein-coupled receptor 4
LGR5leucine rich repeat containing G protein-coupled receptor 5Orphan receptorsAvailableGPR49|FEX|GPR67|orphan G protein-coupled receptor HG38|leucine-rich repeat-containing G protein-coupled receptor 5|leucine-rich repeat containing G protein-coupled receptor 5
LGR6leucine rich repeat containing G protein-coupled receptor 6Orphan receptorsAvailableVTS20631|leucine-rich repeat-containing G protein-coupled receptor 6|leucine-rich repeat containing G protein-coupled receptor 6
MAS1MAS1 proto-oncogene, G protein-coupled receptorOrphan receptorsAvailableMAS|angiotensin 1-7 receptor|MAS1 proto-oncogene, G protein-coupled receptor|MAS1 proto-oncogene
MAS1LMAS1 proto-oncogene like, G protein-coupled receptorOrphan receptorsAvailableMAS-L|MAS-R|MRG
MRGPRDMAS related GPR family member DOrphan receptorsAvailableTGR7|Beta-alanine receptor|G-protein coupled receptor TGR7|mas-related G-protein coupled receptor member D|MAS-related gene D|MAS-related GPR
MRGPREMAS related GPR family member EOrphan receptorsAvailableGPR167|MRGE|MAS-related gene E|MAS-related GPR
MRGPRFMAS related GPR family member FOrphan receptorsAvailableGPR140|GPR168|G-protein coupled receptor 14|MRGF|G-protein coupled receptor RTA|MAS-related gene F|MAS-related GPR
MRGPRGMAS related GPR family member GOrphan receptorsAvailableEBRT2|GPR169|MRGG|MAS-related gene G|MAS-related GPR
MRGPRX1MAS related GPR family member X1Orphan receptorsAvailableMrgc|Mrgprb2|Mrgprc|Mrgprc11|MRGX1|Sensory neuron-specific G-protein coupled receptor 4|SNSR4
MRGPRX2MAS related GPR family member X2Orphan receptorsAvailableMrgprb10|MRGX2
MRGPRX3MAS related GPR family member X3Orphan receptorsAvailableMrgA|Mrgpra|Mrga10|SNSR1|Sensory neuron-specific G protein-coupled receptor 1
MRGPRX4MAS related GPR family member X4Orphan receptorsAvailableSNSR6|MAS-related GPR, member X4|Sensory neuron-specific G-protein coupled receptor 6
TAAR2trace amine associated receptor 2Orphan receptorsAvailableGPR58|G protein-coupled receptor 58|trace amine receptor 2
TAAR5trace amine associated receptor 5Orphan receptorsAvailablePNR|Trace amine receptor 5
TAAR6trace amine associated receptor 6Orphan receptorsAvailableSCZD5|TAR4|Trace amine receptor 4|TRAR4|TA4|trace amine receptor 6
TAAR8trace amine associated receptor 8Orphan receptorsAvailableGPR102|TAR11|TAR5|trace amine receptor 5|trace amine receptor 11|trace amine receptor 8a|trace amine associated receptor 8
TAAR9trace amine associated receptor 9Orphan receptorsAvailableTRAR3|trace amine receptor 3|trace amine receptor 9
GPR143G protein-coupled receptor 143Orphan receptorsAvailableMOA1|ocular albinism 1 (Nettleship-Falls)|NYS6|Ocular albinism type 1 protein
GPR157G protein-coupled receptor 157Orphan receptorsAvailable
GPR156G protein-coupled receptor 156Orphan receptorsAvailablePGR28|PGR22|GABABL|GABAB-related G-protein coupled receptor
GPR158G protein-coupled receptor 158Orphan receptorsAvailable
GPER1G protein-coupled estrogen receptor 1Orphan receptorsAvailableCEPR|CMKRL2|DRY12|FEG-1|Gpr41|LERGU|LERGU2|chemokine receptor-like 2|Flow-induced endothelial G-protein coupled receptor 1|GPGR|LYGPR|Lymphocyte-derived G-protein coupled receptor|Membrane estrogen receptor|mER|GPCR-BR|GPR30|IL8-related receptor DRY12
GPRC5AG protein-coupled receptor class C group 5 member AOrphan receptorsAvailableRAIG1|retinoic acid induced 3|orphan G protein-coupling receptor PEIG-1|retinoic acid-induced gene 1 protein|Retinoic acid-induced protein 3|GPCR5A|RAI3|G protein-coupled receptor, class C, group 5, member A|G protein-coupled receptor
GPRC5BG protein-coupled receptor class C group 5 member BOrphan receptorsAvailableRAIG2|retinoic acid-induced gene 2 protein|G protein-coupled receptor, class C, group 5, member B|G protein-coupled receptor
GPRC5CG protein-coupled receptor class C group 5 member COrphan receptorsAvailableRAIG3|retinoic acid-induced gene 3 protein|G protein-coupled receptor, family C, group 5, member C|G protein-coupled receptor, class C, group 5, member C|G protein-coupled receptor
GPRC5DG protein-coupled receptor class C group 5 member DOrphan receptorsAvailableRAIG4|G protein-coupled receptor, class C, group 5, member D|G protein-coupled receptor
ACKR2atypical chemokine receptor 2Orphan receptorsAvailableCCR10|CCR9|CMBRK9|C-C chemokine receptor D6|chemokine binding protein 2|CMKBR9
ACKR4atypical chemokine receptor 4Orphan receptorsAvailableCC-CKR-11|CCR10|CKR-11|CCR11|PPR1|VSHK1
ACKR1atypical chemokine receptor 1 (Duffy blood group)Orphan receptorsAvailableDuffy antigen/chemokine receptor|atypical chemokine receptor 1|CD234|Dfy|Duffy blood group, atypical chemokine receptor|Darc
GPR176G protein-coupled receptor 176Orphan receptorsAvailableHB954|RBU-15|G-protein coupled receptor AGR9
GPR107G protein-coupled receptor 107Orphan receptorsAvailableLUSTR1|GCDRP|Lung seven transmembrane receptor 1
GPR137G protein-coupled receptor 137Orphan receptorsAvailableGPR137A|TM7SF1L1|TM7SF1|Transmembrane 7 superfamily member 1-like 1 protein
TPRA1transmembrane protein adipocyte associated 1Orphan receptorsAvailableGPR175|TMEM227|TPRA40|G protein-coupled receptor 175|transmembrane protein 227|transmembrane protein, adipocyte asscociated 1|transmembrane protein

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